The antinociceptive actions of dexmedetomidine on dorsal horn neuronal responses in the anaesthetized rat

Eur J Pharmacol. 1992 Apr 29;215(1):127-33. doi: 10.1016/0014-2999(92)90617-d.

Abstract

The actions of the selective alpha 2-adrenoceptor agonist dexmedetomidine were examined on the nociceptive C and innocuous A beta fibre-evoked responses of dorsal horn neurones to transcutaneous electrical stimulation in the intact anaesthetized rat. C fibre-evoked responses were dose dependently reduced by intrathecal dexmedetomidine--to a maximum 86 +/- 6% inhibition by 10 micrograms of the agonist. The ED50 for inhibition of C fibre responses was estimated to be 2.5 micrograms. A beta-evoked responses were inhibited to a lesser degree--a maximum 54 +/- 8% inhibition after 10 micrograms dexmedetomidine. The antinociceptive effects of dexmedetomidine were reversed by the alpha 2-adrenoceptor antagonist atipamezole and the opioid antagonist naloxone. The results are discussed with reference to adrenergic and opioid mechanisms in the spinal cord.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Action Potentials / drug effects
  • Adrenergic alpha-Antagonists / pharmacology
  • Analgesics / antagonists & inhibitors
  • Analgesics / pharmacology*
  • Anesthesia
  • Animals
  • Clonidine / pharmacology
  • Dose-Response Relationship, Drug
  • Electrophysiology
  • Imidazoles / antagonists & inhibitors
  • Imidazoles / pharmacology*
  • Male
  • Medetomidine
  • Naloxone / pharmacology
  • Neurons / drug effects*
  • Neurons / physiology
  • Nociceptors / drug effects*
  • Rats
  • Rats, Inbred Strains
  • Spinal Cord / cytology
  • Spinal Cord / drug effects*
  • Spinal Cord / physiology

Substances

  • Adrenergic alpha-Antagonists
  • Analgesics
  • Imidazoles
  • atipamezole
  • Naloxone
  • Clonidine
  • Medetomidine