Coordination of p300-mediated chromatin remodeling and TRAP/mediator function through coactivator PGC-1alpha

Mol Cell. 2003 Nov;12(5):1137-49. doi: 10.1016/s1097-2765(03)00391-5.

Abstract

Transcriptional coactivators showing physical and functional interactions with PPARgamma include the protein acetyl transferase p300, the TRAP/Mediator complex that interacts with the general transcription machinery, and the highly regulated PGC-1alpha. We show that PGC-1alpha directly interacts with TRAP/Mediator, through the PPARgamma-interacting subunit TRAP220, and stimulates TRAP/Mediator-dependent function on DNA templates. Further, while ineffective by itself, PGC-1alpha stimulates p300-dependent histone acetylation and transcription on chromatin templates in response to PPARgamma. These functions are mediated by largely independent PPARgamma, p300, and TRAP220 interaction domains in PGC-1alpha, whereas p300 and TRAP220 show ligand-dependent interactions with a common region of PPARgamma. Apart from showing PGC-1alpha functions both in chromatin remodeling and in preinitiation complex formation or function (transcription), these results suggest a key role for PGC-1alpha, through concerted but dynamic interactions, in coordinating these steps.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Chromatin / metabolism*
  • E1A-Associated p300 Protein
  • Genes, Reporter
  • HeLa Cells
  • Humans
  • Mediator Complex
  • Mediator Complex Subunit 1
  • Mice
  • Nuclear Proteins / metabolism*
  • Protein Subunits / metabolism
  • Receptors, Cytoplasmic and Nuclear / metabolism
  • Recombinant Fusion Proteins / genetics
  • Recombinant Fusion Proteins / metabolism
  • Trans-Activators / metabolism*
  • Transcription Factors / metabolism*
  • Transcription, Genetic

Substances

  • Chromatin
  • DRIP, VDR interacting protein complex
  • MED1 protein, human
  • MED4 protein, human
  • Med1 protein, mouse
  • Mediator Complex
  • Mediator Complex Subunit 1
  • Nuclear Proteins
  • Protein Subunits
  • Receptors, Cytoplasmic and Nuclear
  • Recombinant Fusion Proteins
  • Trans-Activators
  • Transcription Factors
  • peroxisome-proliferator-activated receptor-gamma coactivator-1
  • E1A-Associated p300 Protein
  • Ep300 protein, mouse