Hypoxia-inducible factor-1-independent regulation of vascular endothelial growth factor by hypoxia in colon cancer

Cancer Res. 2004 Mar 1;64(5):1765-72. doi: 10.1158/0008-5472.can-03-3017.

Abstract

The induction of vascular endothelial growth factor (VEGF) is an essential feature of tumor angiogenesis, and the hypoxia-inducible factor-1 (HIF-1) transcription factor is known to be a key mediator of this process. In colon cancer, the frequently mutated K-ras oncogene also can regulate VEGF expression, but the role that K-ras may play in hypoxia is unknown. Hypoxia induced VEGF promoter activity, mRNA, and protein levels in colon cancer cells. Although HIF-1alpha was induced by hypoxia, VEGF reporter constructs with selectively mutated hypoxia-response elements remained responsive to hypoxia. In addition, "knockdown" of HIF-1alpha by RNA interference only minimally inhibited the hypoxic induction of VEGF. A region of the VEGF promoter between -420 and -90 bp mediated this HIF-independent induction by hypoxia. The introduction of K-ras(Val12) augmented the hypoxic induction of VEGF, and this was observed in wild-type and HIF-1alpha knockdown colon cancer cells. Thus, VEGF may be induced by hypoxia through HIF-dependent and HIF-independent pathways, and K-ras also can induce VEGF in hypoxia independent of HIF-1. These findings suggest the existence of multiple mechanisms regulating the hypoxic induction of VEGF in colon cancer.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Cell Hypoxia*
  • Cell Line, Tumor
  • Colonic Neoplasms / blood supply*
  • DNA-Binding Proteins / physiology*
  • Gene Expression Regulation, Neoplastic*
  • Genes, ras
  • Humans
  • Hypoxia-Inducible Factor 1
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • Neovascularization, Pathologic / etiology
  • Nuclear Proteins / physiology*
  • Promoter Regions, Genetic
  • Transcription Factors*
  • Vascular Endothelial Growth Factor A / genetics*

Substances

  • DNA-Binding Proteins
  • HIF1A protein, human
  • Hypoxia-Inducible Factor 1
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • Nuclear Proteins
  • Transcription Factors
  • Vascular Endothelial Growth Factor A