Fusion of two malaria vaccine candidate antigens enhances product yield, immunogenicity, and antibody-mediated inhibition of parasite growth in vitro

J Immunol. 2004 May 15;172(10):6167-74. doi: 10.4049/jimmunol.172.10.6167.

Abstract

A Plasmodium falciparum chimeric protein 2.9 (PfCP-2.9) was constructed consisting of the C-terminal regions of two leading malaria vaccine candidates, domain III of apical membrane ag-1 (AMA-1) and 19-kDa C-terminal fragment of the merozoite surface protein 1 (MSP1). The PfCP-2.9 was produced by Pichia pastoris in secreted form with a yield of 2600 mg/L and approximately 1 g/L of final product was obtained from a three-step purification process. Analysis of conformational properties of the chimeric protein showed that all six conformational mAbs interacted with the recombinant protein were reduction-sensitive, indicating that fusion of the two cysteine-rich proteins retains critical conformational epitopes. PfCP-2.9 was found to be highly immunogenic in rabbits as well as in rhesus monkeys (Macaca mulatta). The chimeric protein induced both anti-MSP1-19 and anti-AMA-1(III) Abs at levels 11- and 18-fold higher, respectively, than individual components did. Anti-PfCP-2.9 sera from both rabbits and rhesus monkeys almost completely inhibited in vitro growth of the P. falciparum FCC1/HN and 3D7 lines when tested at a 6.7-fold dilution. It was shown that the inhibition is dependent on the presence of Abs to the chimeric protein and their disulfide bond-dependent conformations. Moreover, the activity was mediated by a combination of growth-inhibitory Abs generated by the individual MSP1-19 and AMA-1(III) of PfCP-2.9. The combination of the extremely high yield of the protein and enhancement of its immune response provides a basis to develop an effective and affordable malaria vaccine.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adjuvants, Immunologic / administration & dosage
  • Adjuvants, Immunologic / chemical synthesis
  • Adjuvants, Immunologic / genetics
  • Animals
  • Antibodies, Protozoan / physiology*
  • Antigens, Protozoan / administration & dosage
  • Antigens, Protozoan / genetics*
  • Antigens, Protozoan / immunology
  • Antiprotozoal Agents / administration & dosage
  • Antiprotozoal Agents / chemical synthesis
  • Antiprotozoal Agents / immunology*
  • Calcium-Binding Proteins / administration & dosage
  • Calcium-Binding Proteins / genetics*
  • Calcium-Binding Proteins / immunology
  • Growth Inhibitors / administration & dosage
  • Growth Inhibitors / chemical synthesis
  • Growth Inhibitors / genetics
  • Growth Inhibitors / immunology
  • Macaca mulatta
  • Malaria Vaccines / administration & dosage
  • Malaria Vaccines / chemical synthesis
  • Malaria Vaccines / genetics*
  • Malaria Vaccines / immunology
  • Membrane Proteins / administration & dosage
  • Membrane Proteins / genetics*
  • Membrane Proteins / immunology
  • Molecular Sequence Data
  • Plasmodium falciparum / growth & development*
  • Plasmodium falciparum / immunology
  • Protein Kinases / administration & dosage
  • Protein Kinases / genetics*
  • Protein Kinases / immunology
  • Protozoan Proteins / administration & dosage
  • Protozoan Proteins / genetics*
  • Protozoan Proteins / immunology
  • Rabbits
  • Recombinant Fusion Proteins / administration & dosage
  • Recombinant Fusion Proteins / chemical synthesis
  • Recombinant Fusion Proteins / genetics*
  • Recombinant Fusion Proteins / immunology
  • Subtilisins / administration & dosage
  • Subtilisins / genetics
  • Subtilisins / immunology
  • Vaccines, DNA / administration & dosage
  • Vaccines, DNA / chemical synthesis
  • Vaccines, DNA / immunology*

Substances

  • Adjuvants, Immunologic
  • Antibodies, Protozoan
  • Antigens, Protozoan
  • Antiprotozoal Agents
  • Calcium-Binding Proteins
  • Growth Inhibitors
  • Malaria Vaccines
  • Membrane Proteins
  • Protozoan Proteins
  • Recombinant Fusion Proteins
  • Vaccines, DNA
  • apical membrane antigen I, Plasmodium
  • Protein Kinases
  • PfCPK protein, Plasmodium falciparum
  • Subtilisins
  • sub-2 protein, Plasmodium falciparum

Associated data

  • GENBANK/AY496866