Budesonide/formoterol combination therapy as both maintenance and reliever medication in asthma

Am J Respir Crit Care Med. 2005 Jan 15;171(2):129-36. doi: 10.1164/rccm.200407-884OC. Epub 2004 Oct 22.

Abstract

Asthma control is improved by combining inhaled corticosteroids with long-acting beta2-agonists. However, fluctuating asthma control still occurs. We hypothesized that in patients receiving low maintenance dose budesonide/formoterol (bud/form), replacing short-acting beta2-agonist (SABA) reliever with as-needed bud/form would provide rapid symptom relief and simultaneous adjustment in antiinflammatory therapy, thereby reducing exacerbations. In this double-blind, randomized, parallel-group study, 2,760 patients with asthma aged 4-80 years (FEV1 60-100% predicted) received either terbutaline 0.4 mg as SABA with bud/form 80/4.5 microg twice a day (bud/form + SABA) or bud 320 microg twice a day (bud + SABA) or bud/form 80/4.5 microg twice a day with 80/4.5 microg as-needed (bud/form maintenance + relief). Children used a once-nocte maintenance dose. Bud/form maintenance + relief prolonged time to first severe exacerbation (p < 0.001; primary endpoint), resulting in a 45-47% lower exacerbation risk versus bud/form + SABA (hazard ratio, 0.55; 95% confidence interval, 0.44, 0.67) or bud + SABA (hazard ratio, 0.53; 95% confidence interval 0.43, 0.65). Bud/form maintenance + relief also prolonged the time to the first, second, and third exacerbation requiring medical intervention (p < 0.001), reduced severe exacerbation rate, and improved symptoms, awakenings, and lung function compared with both fixed dosing regimens.

Publication types

  • Clinical Trial
  • Multicenter Study
  • Randomized Controlled Trial

MeSH terms

  • Adolescent
  • Adrenergic beta-Agonists / administration & dosage*
  • Adrenergic beta-Agonists / adverse effects
  • Adrenergic beta-Agonists / pharmacology
  • Adult
  • Aged
  • Aged, 80 and over
  • Anti-Inflammatory Agents / administration & dosage*
  • Anti-Inflammatory Agents / adverse effects
  • Anti-Inflammatory Agents / pharmacology
  • Asthma / drug therapy*
  • Budesonide / administration & dosage*
  • Budesonide / adverse effects
  • Budesonide / pharmacology
  • Child
  • Child, Preschool
  • Double-Blind Method
  • Drug Combinations
  • Ethanolamines / administration & dosage*
  • Ethanolamines / adverse effects
  • Ethanolamines / pharmacology
  • Female
  • Formoterol Fumarate
  • Humans
  • Male
  • Metered Dose Inhalers
  • Middle Aged
  • Peak Expiratory Flow Rate / drug effects
  • Proportional Hazards Models
  • Regression Analysis
  • Safety

Substances

  • Adrenergic beta-Agonists
  • Anti-Inflammatory Agents
  • Drug Combinations
  • Ethanolamines
  • Budesonide
  • Formoterol Fumarate