DNA-PKcs, but not TLR9, is required for activation of Akt by CpG-DNA

EMBO J. 2005 Feb 23;24(4):779-89. doi: 10.1038/sj.emboj.7600539. Epub 2005 Jan 27.

Abstract

CpG-DNA and its related synthetic CpG oligodeoxynucleotides (CpG-ODNs) play an important role in immune cell survival. It has been suggested that Akt is one of the CpG-DNA-responsive serine/threonine kinases; however, the target protein of CpG-DNA that leads to Akt activation has not been elucidated. Here, we report that ex vivo stimulation of bone marrow-derived macrophages (BMDMs) from mice lacking the catalytic subunit of DNA-dependent protein kinase (DNA-PKcs) results in defective phosphorylation and activation of Akt by CpG-DNA. Unexpectedly, loss of the Toll-like receptor 9 has a minimal effect on Akt activation in response to CpG-DNA. Further in vitro analysis using purified DNA-PK and recombinant Akt proteins reveals that DNA-PK directly induces phosphorylation and activation of Akt. In addition, in BMDMs, DNA-PKcs associates with Akt upon CpG-DNA stimulation and triggers transient nuclear translocation of Akt. Thus, our findings establish a novel role for DNA-PKcs in CpG-DNA signaling and define a CpG-DNA/DNA-PKcs/Akt pathway.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Active Transport, Cell Nucleus / drug effects
  • Animals
  • Bone Marrow / drug effects
  • Bone Marrow / enzymology
  • Cells, Cultured
  • DNA-Activated Protein Kinase
  • DNA-Binding Proteins / metabolism*
  • Enzyme Activation
  • Macrophages / drug effects
  • Macrophages / enzymology
  • Mice
  • Mice, Knockout
  • Oligodeoxyribonucleotides / pharmacology*
  • Phosphorylation
  • Protein Serine-Threonine Kinases / metabolism*
  • Proto-Oncogene Proteins / metabolism*
  • Proto-Oncogene Proteins c-akt
  • Receptors, Cell Surface / metabolism
  • Toll-Like Receptor 9

Substances

  • CPG-oligonucleotide
  • DNA-Binding Proteins
  • Oligodeoxyribonucleotides
  • Proto-Oncogene Proteins
  • Receptors, Cell Surface
  • Tlr9 protein, mouse
  • Toll-Like Receptor 9
  • DNA-Activated Protein Kinase
  • Protein Serine-Threonine Kinases
  • Proto-Oncogene Proteins c-akt