Dihydrodiol dehydrogenase activities of rabbit liver are associated with hydroxysteroid dehydrogenases and aldo-keto reductases

Eur J Biochem. 1992 May 1;205(3):1155-62. doi: 10.1111/j.1432-1033.1992.tb16885.x.

Abstract

1. Dihydrodiol dehydrogenase activities were investigated in rabbit liver. Using a five-step purification scheme, eight isoenzymes of dihydrodiol dehydrogenase with isoelectric points of 5.55-9.3 and promoter molecular masses of 34-35 kDa were purified to apparent homogeneity and designated CF-1 to CF-6, CM-1 and CM-2. 2. CF-1 and CF-2 had near-neutral isoelectric points of 7.4 and 6.8 and molecular masses of about 125 kDa in the native state. Both enzymes readily accepted NAD+ as well as NADP+ as coenzymes, had relatively low Km values of 0.33 mM and 0.47 mM for benzene dihydrodiol and resembled previously described carbonyl reductases in their substrate specificity towards ketones and quinones. 3. CF-5 and CF-6 had acidic isoelectric points of 5.9 and 5.55 and native molecular masses of approximately 60 kDa. They displayed a strong preference for NADP(H) as coenzyme and had high Km and Vmax with benzene dihydrodiol. Since these enzymes reduced p-nitrobenzaldehyde and glucuronic acid efficiently, they appeared to be closely related to aldehyde reductase. 4. CF-4 had a high 3 alpha-hydroxysteroid dehydrogenase activity for the diagnostic substrate androsterone, a moderate activity for other 3 alpha-hydroxysteroids as well as 17 alpha-hydroxysteroids, and relatively low activities for 3 beta-hydroxysteroids and 17 beta-hydroxysteroids. CF-5 and CM-1 had high 17 beta-hydroxysteroid dehydrogenase activity for the diagnostic substrate 5 alpha-dihydrotestosterone, and low to moderate activities for other 17 beta-hydroxysteroids as well as 3 alpha-hydroxysteroids. 5. The isoenzyme CM-2 had an isoelectric point of 9.3 and was a very active quinone reductase with phenanthrene-9,10-quinone as substrate. It was potently inhibited by phenobarbital. 6. We conclude that the dihydrodiol dehydrogenase activities of rabbit liver are associated with aldehyde and carbonyl reductase and with 3 alpha-hydroxysteroid and 17 beta-hydroxysteroid dehydrogenases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alcohol Oxidoreductases / isolation & purification
  • Alcohol Oxidoreductases / metabolism*
  • Aldehyde Reductase
  • Aldo-Keto Reductases
  • Animals
  • Antibodies, Monoclonal
  • Catalysis
  • Electrophoresis, Polyacrylamide Gel
  • Hydroxysteroid Dehydrogenases / metabolism*
  • Isoelectric Point
  • Isoenzymes / isolation & purification
  • Isoenzymes / metabolism*
  • Liver / enzymology*
  • Male
  • Molecular Weight
  • Oxidoreductases Acting on CH-CH Group Donors*
  • Oxidoreductases*
  • Rabbits
  • Substrate Specificity
  • Tissue Distribution

Substances

  • Antibodies, Monoclonal
  • Isoenzymes
  • Oxidoreductases
  • Alcohol Oxidoreductases
  • Hydroxysteroid Dehydrogenases
  • dihydrodiol dehydrogenases
  • Aldo-Keto Reductases
  • Aldehyde Reductase
  • Oxidoreductases Acting on CH-CH Group Donors
  • cis-1,2-dihydro-1,2-dihydroxynaphthalene dehydrogenase