Phase II study of celecoxib in metastatic differentiated thyroid carcinoma

J Clin Endocrinol Metab. 2006 Jun;91(6):2201-4. doi: 10.1210/jc.2005-2498. Epub 2006 Mar 7.

Abstract

Context: There is increased cyclooxygenase-2 (COX-2) expression in malignant thyroid nodules compared with nonneoplastic and benign thyroid tissue.

Objective: The objective of the study was to evaluate the efficacy of celecoxib, a selective COX-2 inhibitor, in treating patients with progressive metastatic differentiated thyroid cancer (DTC) and to explore the relationship of clinical response to tumor COX-2 expression with immunohistochemistry in a subset of patients.

Design: The study was a prospective phase II trial with Fleming single-stage design powered at 80% with a 5% rejection error to detect more than 20% progression-free survival at 12 months.

Setting: Ambulatory patients were from tertiary referral academic medical centers.

Patients: Patients in the study had progressive metastatic DTC and had failed prior standard therapy.

Intervention: Patients were treated with celecoxib 400 mg orally twice a day for 12 months.

Main outcome measure: The main outcome measure was progression-free survival at 12 months of treatment using Response Evaluation Criteria in Solid Tumors and/or serum thyroglobulin.

Results: Twenty-three of 32 patients experienced progressive disease or stopped therapy due to toxicity, thus fulfilling the intent-to-treat study endpoint for celecoxib failure. One patient achieved partial response, and one patient completed 12 months of therapy progression-free. The patient with partial response was on therapy along with seven other patients when the study was terminated.

Conclusions: Celecoxib 400 mg orally twice per day fails to halt progressive metastatic DTC in most patients.

Publication types

  • Clinical Trial, Phase II
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Celecoxib
  • Cyclooxygenase 2 / analysis
  • Cyclooxygenase 2 Inhibitors / therapeutic use*
  • Female
  • Humans
  • Male
  • Middle Aged
  • Prospective Studies
  • Pyrazoles / adverse effects
  • Pyrazoles / therapeutic use*
  • Sulfonamides / adverse effects
  • Sulfonamides / therapeutic use*
  • Thyroid Neoplasms / drug therapy*
  • Thyroid Neoplasms / enzymology

Substances

  • Cyclooxygenase 2 Inhibitors
  • Pyrazoles
  • Sulfonamides
  • Cyclooxygenase 2
  • Celecoxib