Comparison of putative cGMP-binding regions in bovine brain and cardiac cGMP-stimulated phosphodiesterases

Second Messengers Phosphoproteins. 1991;13(2-3):87-98.

Abstract

After photolabelling of purified bovine brain particulate cGMP stimulated phosphodiesterase (PDE) with [32P]cGMP, incubation with V8 Endoproteinase Glu-C produced several fragments; most of the [32P] was associated with smaller fragments (approximately 12-14 kDa), and some occasionally with larger fragments (approximately 55-57 kDa). Partial amino acid sequences were determined for the smaller photolabelled fragments and other peptides. On Western immunoblots, affinity-purified antibodies against a synthetic peptide with a sequence matching part of that of the approximately 12-14 kDa photolabelled material reacted with intact PDE and the approximately 12-14 kDa and approximately 55-57 kDa fragments. Several partial cDNA clones encoding the cGMP-stimulated PDE were isolated from a Lambda Zap II bovine brain cDNA library. Deduced amino acid sequence from one cDNA clone, lambda cGS 3-1, as well as the partial sequence of the approximately 12-14 kDa and other fragments, exhibited considerable identity with amino acid residues 311-921 of the cardiac cGMP-stimulated PDE (Trong et al., 1990), including the putative cGMP-binding domain (Charbonneau et al., 1990). These results further define this cGMP-binding domain and suggest that different cGMP-stimulated PDEs will exhibit considerable homology, at least in their cGMP-binding region(s) and catalytic domains.

Publication types

  • Comparative Study

MeSH terms

  • 3',5'-Cyclic-GMP Phosphodiesterases / genetics
  • 3',5'-Cyclic-GMP Phosphodiesterases / immunology
  • 3',5'-Cyclic-GMP Phosphodiesterases / isolation & purification*
  • Affinity Labels
  • Amino Acid Sequence
  • Animals
  • Base Sequence
  • Binding Sites
  • Blotting, Western
  • Brain / enzymology*
  • Cattle
  • Cyclic GMP / isolation & purification*
  • DNA / genetics
  • DNA / isolation & purification
  • Electrophoresis, Polyacrylamide Gel
  • Male
  • Molecular Sequence Data
  • Myocardium / enzymology*
  • Oligonucleotide Probes
  • Oligopeptides / chemical synthesis
  • Oligopeptides / genetics
  • Oligopeptides / immunology
  • Peptide Fragments
  • Rabbits

Substances

  • Affinity Labels
  • Oligonucleotide Probes
  • Oligopeptides
  • Peptide Fragments
  • DNA
  • 3',5'-Cyclic-GMP Phosphodiesterases
  • Cyclic GMP