Distinct role of the N-terminal tail of the Na,K-ATPase catalytic subunit as a signal transducer

J Biol Chem. 2006 Aug 4;281(31):21954-21962. doi: 10.1074/jbc.M601578200. Epub 2006 May 24.

Abstract

Mounting evidence suggests that the ion pump, Na,K-ATPase, can, in the presence of ouabain, act as a signal transducer. A prominent binding motif linking the Na,K-ATPase to intracellular signaling effectors has, however, not yet been identified. Here we report that the N-terminal tail of the Na,K-ATPase catalytic alpha-subunit (alphaNT-t) binds directly to the N terminus of the inositol 1,4,5-trisphosphate receptor. Three amino acid residues, LKK, conserved in most species and most alpha-isoforms, are essential for the binding to occur. In wild-type cells, low concentrations of ouabain trigger low frequency calcium oscillations that activate NF-kappaB and protect from apoptosis. All of these effects are suppressed in cells overexpressing a peptide corresponding to alphaNT-t but not in cells overexpressing a peptide corresponding to alphaNT-t deltaLKK. Thus we have identified a well conserved Na,K-ATPase motif that binds to the inositol 1,4,5-trisphosphate receptor and can trigger an anti-apoptotic calcium signal.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis
  • Binding Sites
  • Calcium Channels / metabolism
  • Calcium Signaling
  • Catalysis
  • Humans
  • Inositol 1,4,5-Trisphosphate Receptors
  • Male
  • Membrane Glycoproteins / metabolism
  • Mice
  • NF-kappa B / metabolism
  • Ouabain / pharmacology
  • Protein Binding
  • Protein Subunits / metabolism
  • Protein Subunits / physiology
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Cytoplasmic and Nuclear / metabolism
  • Signal Transduction*
  • Sodium-Potassium-Exchanging ATPase / chemistry
  • Sodium-Potassium-Exchanging ATPase / metabolism
  • Sodium-Potassium-Exchanging ATPase / physiology*

Substances

  • Calcium Channels
  • Inositol 1,4,5-Trisphosphate Receptors
  • Itpr1 protein, mouse
  • Membrane Glycoproteins
  • NF-kappa B
  • Protein Subunits
  • Receptors, Cytoplasmic and Nuclear
  • Ouabain
  • ATP1A1 protein, human
  • Atp1a1 protein, rat
  • Atp1a1 protein, mouse
  • Sodium-Potassium-Exchanging ATPase