Rac1 links integrin-mediated adhesion to the control of lactational differentiation in mammary epithelia

J Cell Biol. 2006 Jun 5;173(5):781-93. doi: 10.1083/jcb.200601059.

Abstract

The expression of tissue-specific genes during mammary gland differentiation relies on the coincidence of two distinct signaling events: the continued engagement of beta1 integrins with the extracellular matrix (ECM) and a hormonal stimulus from prolactin (Prl). How the integrin and Prl receptor (PrlR) systems integrate to regulate milk protein gene synthesis is unknown. In this study, we identify Rac1 as a key link. Dominant-negative Rac1 prevents Prl-induced synthesis of the milk protein beta-casein in primary mammary epithelial cells cultured as three-dimensional acini on basement membrane. Conversely, activated Rac1 rescues the defective beta-casein synthesis that occurs under conditions not normally permissive for mammary differentiation, either in beta1 integrin-null cells or in wild-type cells cultured on collagen. Rac1 is required downstream of integrins for activation of the PrlR/Stat5 signaling cascade. Cdc42 is also necessary for milk protein synthesis but functions via a distinct mechanism to Rac1. This study identifies the integration of signals provided by ECM and hormones as a novel role for Rho family guanosine triphosphatases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Caseins / biosynthesis
  • Caseins / drug effects
  • Cell Adhesion / physiology
  • Cell Differentiation / physiology
  • Cells, Cultured
  • Epithelial Cells / metabolism
  • Epithelial Cells / physiology*
  • Extracellular Matrix / physiology
  • Female
  • GTP Phosphohydrolases / physiology
  • GTPase-Activating Proteins / drug effects
  • GTPase-Activating Proteins / pharmacology
  • GTPase-Activating Proteins / physiology
  • Integrin beta1 / metabolism*
  • Lactation / metabolism*
  • Mammary Glands, Animal / physiology
  • Mice
  • Mice, Inbred ICR
  • Neuropeptides / metabolism*
  • Neuropeptides / pharmacology
  • Pregnancy
  • Prolactin / antagonists & inhibitors
  • Prolactin / pharmacology
  • Signal Transduction / physiology
  • rac GTP-Binding Proteins / metabolism*
  • rac GTP-Binding Proteins / pharmacology
  • rac1 GTP-Binding Protein

Substances

  • Arhgap31 protein, mouse
  • Caseins
  • GTPase-Activating Proteins
  • Integrin beta1
  • Neuropeptides
  • Rac1 protein, mouse
  • Prolactin
  • GTP Phosphohydrolases
  • rac GTP-Binding Proteins
  • rac1 GTP-Binding Protein