Novel nucleotide triphosphates as potent P2Y2 agonists

Bioorg Med Chem Lett. 2007 Jan 15;17(2):562-5. doi: 10.1016/j.bmcl.2006.09.017. Epub 2006 Sep 29.

Abstract

The synthesis and P2Y2 activities of a novel series of nucleoside triphosphates are described. Many of these compounds were potent agonists of the P2Y2 receptor.

Publication types

  • Comparative Study

MeSH terms

  • Cell Line, Tumor
  • DNA, Complementary / biosynthesis
  • DNA, Complementary / genetics
  • Humans
  • Indicators and Reagents
  • Magnetic Resonance Spectroscopy
  • Nucleotides / chemical synthesis*
  • Nucleotides / pharmacology*
  • Purinergic P2 Receptor Agonists*
  • Receptors, Purinergic P2Y2
  • Reverse Transcriptase Polymerase Chain Reaction
  • Structure-Activity Relationship
  • Uridine Triphosphate / pharmacology

Substances

  • DNA, Complementary
  • Indicators and Reagents
  • Nucleotides
  • P2RY2 protein, human
  • Purinergic P2 Receptor Agonists
  • Receptors, Purinergic P2Y2
  • Uridine Triphosphate