A novel hepatitis B virus mutation with resistance to adefovir but not to tenofovir in an HIV-hepatitis B virus-co-infected patient

AIDS. 2006 Nov 14;20(17):2229-31. doi: 10.1097/01.aids.0000252061.35422.84.

Abstract

A molecular virology analysis performed in an HIV-hepatitis B virus (HBV) co-infected patient showed the emergence of an unusual HBV polymerase gene mutation (rt A181T) under adefovir therapy, conferring resistance to adefovir but not to tenofovir, as proved by in-vitro phenotypic analysis. This observation suggests that careful monitoring of co-infected patients is required to diagnose HBV resistance to nucleos(t)ide analogues, and that tenofovir may be active at least against some of the adefovir-resistant strains.

Publication types

  • Case Reports
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenine / analogs & derivatives
  • Adenine / therapeutic use
  • Adult
  • Drug Resistance, Viral
  • Gene Products, pol / genetics*
  • HIV Infections / complications*
  • Hepatitis B virus / genetics*
  • Hepatitis B, Chronic / complications
  • Hepatitis B, Chronic / drug therapy*
  • Humans
  • Mutation / genetics*
  • Organophosphonates / therapeutic use
  • Reverse Transcriptase Inhibitors / therapeutic use*
  • Tenofovir

Substances

  • Gene Products, pol
  • Organophosphonates
  • P protein, Hepatitis B virus
  • Reverse Transcriptase Inhibitors
  • adefovir
  • Tenofovir
  • Adenine