Phase II trial of gemcitabine, prednisone, and zoledronic acid in pretreated patients with hormone refractory prostate cancer

Urology. 2007 Feb;69(2):347-51. doi: 10.1016/j.urology.2006.10.007.

Abstract

Objectives: To investigate the impact on biochemical and objective response and on pain improvement of gemcitabine, prednisone, and zoledronic acid in patients with hormone-refractory prostate cancer (HRPC), previously treated with docetaxel-based regimens.

Methods: The patients were treated with gemcitabine 1000 mg/m2 every 14 days, prednisone 10 mg orally on days 1 to 7 and 14 to 21, and zoledronic acid every 4 weeks. Changes in prostate-specific antigen levels, tumor response, and toxicity were evaluated every month. The pain response, based on pain reduction and analgesic drug reduction, was assessed during therapy.

Results: A total of 22 men (median age 65 years) were treated. Overall, 5 patients (23%) achieved a 50% or greater reduction in prostate-specific antigen level after two cycles; a partial response was observed in 1 (14%) of 7 patients with measurable disease, and 3 (43%) of 7 had stable disease. Of the 22 men, 23% had pain improvement. The most important hematologic toxicity was neutropenia (grade 3 in 18%).

Conclusions: The combination of gemcitabine, prednisone, and zoledronic acid appears to be associated with biochemical response, pain improvement, and good safety in pretreated patients with HRPC.

Publication types

  • Clinical Trial, Phase II

MeSH terms

  • Aged
  • Aged, 80 and over
  • Antineoplastic Combined Chemotherapy Protocols / administration & dosage*
  • Deoxycytidine / administration & dosage
  • Deoxycytidine / analogs & derivatives
  • Diphosphonates / administration & dosage
  • Dose-Response Relationship, Drug
  • Drug Administration Schedule
  • Drug Resistance, Neoplasm
  • Follow-Up Studies
  • Gemcitabine
  • Humans
  • Imidazoles / administration & dosage
  • Male
  • Middle Aged
  • Neoplasm Invasiveness / pathology
  • Neoplasm Staging
  • Neoplasms, Hormone-Dependent
  • Pain Measurement
  • Palliative Care*
  • Prednisone / administration & dosage
  • Probability
  • Prostate-Specific Antigen / blood
  • Prostate-Specific Antigen / drug effects*
  • Prostatic Neoplasms / drug therapy*
  • Prostatic Neoplasms / mortality*
  • Prostatic Neoplasms / pathology
  • Risk Assessment
  • Survival Rate
  • Treatment Outcome
  • Zoledronic Acid

Substances

  • Diphosphonates
  • Imidazoles
  • Deoxycytidine
  • Zoledronic Acid
  • Prostate-Specific Antigen
  • Prednisone
  • Gemcitabine