Induction of uterine calbindin-D9k through an estrogen receptor-dependent pathway following single injection with xenobiotic agents in immature rats

J Toxicol Environ Health A. 2007 Jan 15;70(2):171-82. doi: 10.1080/15287390600755257.

Abstract

Various environmental chemicals, both natural and synthetic, are believed to act as endocrine disruptors (EDs) in mammals. In this study, a new in vivo model of immature rats was used to explore the induction of calbindin-D9k (CaBP-9k) following a single injection of EDs. In a time-dependent experiment, immature rats at postnatal day 16 were treated with high doses (600 mg/kg body weight [BW]) of 4-tert-octyphenol (OP), p-nonylphenol (NP), or bisphenol A (BPA), and euthanized at different time points (3, 6, 12, 24, or 48 h). For a dose-dependent study, immature rats were given different doses (200, 400, or 600 mg/kg BW) and euthanized at 24 h after injection. After treatment with these EDs, the effects on CaBP-9k mRNA and protein were examined by Northern and Western blot analyses, respectively. An anti-estrogen, ICI 182,780, was employed to examine the potential involvement of estrogen receptor (ER) in the induction of estrogen receptor-mediated physiologic responses in vivo. A single treatment with each of the chemicals, at 600 mg/kg BW, resulted in a significant increase in the expression of CaBP-9k mRNA and protein 24 h after injection. In addition, treatment with OP, NP, or BPA resulted in a positive uterotrophic response. Cotreatment with the ER antagonist ICI 182,780 completely prevented the ED-induced uterine weight gain. Taken together, these results demonstrate that a single injection of OP, NP, or BPA results in an increase of CaBP-9k mRNA and protein via an ER-dependent pathway in the uterus of immature rats. This new model may be important to elucidate the mechanism of action of xenoestrogens on estrogen-sensitive tissue.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Benzhydryl Compounds
  • Calbindins
  • Endocrine Disruptors / toxicity
  • Estradiol / analogs & derivatives
  • Estradiol / pharmacology
  • Estrogen Antagonists / pharmacology
  • Estrogens, Non-Steroidal / toxicity
  • Female
  • Fulvestrant
  • Injections, Subcutaneous
  • Organ Size / drug effects
  • Phenols / toxicity*
  • RNA, Messenger / biosynthesis
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Estrogen / antagonists & inhibitors
  • Receptors, Estrogen / metabolism
  • S100 Calcium Binding Protein G / biosynthesis*
  • S100 Calcium Binding Protein G / genetics
  • Uterus / drug effects*
  • Uterus / growth & development
  • Uterus / metabolism
  • Xenobiotics / toxicity

Substances

  • Benzhydryl Compounds
  • Calbindins
  • Endocrine Disruptors
  • Estrogen Antagonists
  • Estrogens, Non-Steroidal
  • Phenols
  • RNA, Messenger
  • Receptors, Estrogen
  • S100 Calcium Binding Protein G
  • S100g protein, rat
  • Xenobiotics
  • Fulvestrant
  • Estradiol
  • nonylphenol
  • 4-tert-octylphenol
  • bisphenol A