p53 and SCFFbw7 cooperatively restrain cyclin E-associated genome instability

Oncogene. 2007 Oct 18;26(48):6948-53. doi: 10.1038/sj.onc.1210518. Epub 2007 May 7.

Abstract

Cancers often exhibit high levels of cyclin E expression, and aberrant cyclin E activity causes genomic instability and increased tumorigenesis. Two tumor suppressor pathways protect cells against cyclin E deregulation. The p53 pathway is induced by excess cyclin E in primary cells and opposes cyclin E activity through induction of p21Cip1. In contrast, the Fbw7 pathway targets cyclin E for degradation, and Fbw7 mutations occur commonly in cancers. We investigated the cooperativity of these two pathways in countering cyclin E-induced genomic instability in primary human cells. We find that loss of p53 and Fbw7 synergistically unmasks cyclin E-induced instability. In normal cells, impaired cyclin E degradation produces genome instability, but this is rapidly mitigated by induction of p53 and p21. In contrast, p53 loss allows the high level of cyclin E kinase activity that results from Fbw7 loss to persist and continuously drive genome instability. Moreover, p21 plays a critical role in suppressing cyclin E when Fbw7 is disabled, and in the absence of p21, sustained cyclin E activity induces rapid cell death via apoptosis. These data directly demonstrate the cooperative roles of these Fbw7 and p53 pathways in restraining cyclin E activity and its associated genome instability.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Apoptosis
  • Cyclin E / genetics
  • Cyclin E / metabolism*
  • Fibroblasts / cytology
  • Fibroblasts / metabolism*
  • Genomic Instability
  • Humans
  • Immunoblotting
  • Immunoprecipitation
  • Micronucleus Tests
  • Oncogene Proteins / genetics
  • Oncogene Proteins / metabolism*
  • Poly(ADP-ribose) Polymerases / metabolism
  • SKP Cullin F-Box Protein Ligases / antagonists & inhibitors
  • SKP Cullin F-Box Protein Ligases / genetics
  • SKP Cullin F-Box Protein Ligases / metabolism*
  • Tumor Suppressor Protein p53 / genetics
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • CCNE1 protein, human
  • Cyclin E
  • Oncogene Proteins
  • Tumor Suppressor Protein p53
  • SKP Cullin F-Box Protein Ligases
  • Poly(ADP-ribose) Polymerases