Chronic AT1-receptor blockade does not alter cerebral oxygen supply/demand ratio during cardiopulmonary bypass in hypertensive patients

Acta Anaesthesiol Scand. 2008 Jan;52(1):73-80. doi: 10.1111/j.1399-6576.2007.01479.x. Epub 2007 Nov 1.

Abstract

Background: The angiotensin II receptor type 1 antagonist candesartan has been hypothesized to alter vasopressor requirements and brain-blood flow by changing cerebrovascular autoregulation. Therefore, we assessed the effects of a pre-anaesthetic treatment course with candesartan on cerebral arterial-jugular bulb oxygen content difference, middle cerebral artery blood velocity, and vasopressor requirements in hypertensive patients undergoing elective on-pump coronary artery bypass graft surgery.

Methods: In a randomized, double-blind, placebo-controlled study, we evaluated the effects of candesartan (8 mg po/d, given for 6-8 days before surgery) in 35 hypertensive patients. The mean arterial pressure was maintained above 60 mmHg by bolus administration of phenylephrine, if required, and dosages were recorded.

Results: Candesartan did not significantly alter oxygen content difference across the cerebral circulation, mean middle cerebral artery blood velocity during cardiopulmonary bypass, or phenylephrine requirements either before (0.0067 microg/kg/min+/-0.0042 vs. 0.0056 microg/kg/min+/-0.0049, P=0.48) or during cardiopulmonary bypass (0.0240 microg/kg/min+/-0.0240 vs. 0.0250 microg/kg/min+/-0.0190, P=0.97) compared with placebo.

Conclusion: Thus, a 6-8-day treatment course with candesartan does not alter global cerebral perfusion and oxygen supply/demand ratio during cardiopulmonary bypass, or vasopressor requirements in hypertensive patients undergoing on-pump coronary artery bypass graft surgery, and no deleterious consequences of AT1-receptor blockade were detected.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Aged
  • Angiotensin II Type 1 Receptor Blockers / pharmacology*
  • Angiotensin II Type 1 Receptor Blockers / therapeutic use
  • Antihypertensive Agents / pharmacology*
  • Antihypertensive Agents / therapeutic use
  • Benzimidazoles / pharmacology*
  • Benzimidazoles / therapeutic use
  • Biphenyl Compounds
  • Blood Flow Velocity / drug effects
  • Blood Pressure / drug effects
  • Brain / metabolism*
  • Cardiopulmonary Bypass* / adverse effects
  • Cerebral Arteries
  • Cerebrovascular Circulation / drug effects*
  • Double-Blind Method
  • Female
  • Humans
  • Hypertension / complications
  • Hypertension / drug therapy*
  • Hypoxia, Brain / etiology
  • Hypoxia, Brain / prevention & control*
  • Intraoperative Complications / etiology
  • Intraoperative Complications / prevention & control*
  • Jugular Veins
  • Male
  • Middle Aged
  • Middle Cerebral Artery
  • Oxygen / metabolism*
  • Phenylephrine / administration & dosage
  • Phenylephrine / therapeutic use
  • Premedication
  • Tetrazoles / pharmacology*
  • Tetrazoles / therapeutic use
  • Treatment Failure

Substances

  • Angiotensin II Type 1 Receptor Blockers
  • Antihypertensive Agents
  • Benzimidazoles
  • Biphenyl Compounds
  • Tetrazoles
  • Phenylephrine
  • Oxygen
  • candesartan