Hepatotoxicity of nevirapine in virologically suppressed patients according to gender and CD4 cell counts

HIV Med. 2008 Apr;9(4):221-6. doi: 10.1111/j.1468-1293.2008.00552.x.

Abstract

Objectives: A warning advising a higher risk of hepatotoxicity in antiretroviral-naive patients starting a nevirapine-containing combination antiretroviral therapy (NcART) has been issued by health authorities. It is unclear whether this higher risk also applies to stable virologically suppressed patients starting NcART.

Methods: We performed a meta-analysis of published randomized studies including virologically suppressed patients who switched to NcART with a follow-up >or=3 months. CD4 cell cell counts were classified as high (HCD4) (400 cells/microL for males and 250 cells/microL for females) or low (LCD4). The main endpoint was hepatotoxicity within the first 3 months.

Results: Four studies with a pooled total of 410 patients were included. The risk of hepatotoxicity within the first 3 months was 2% and 4% in the LCD4 and HCD4 groups, respectively, with a combined odds ratio of 1.46 [95% confidence interval (CI) 0.43-4.98; P=0.54]. The risk of hepatotoxicity at any point during the study was similar in both groups, with a combined hazard ratio of 0.8 (95% CI 0.3-2.5; P=0.80).

Conclusions: In our study, virologically suppressed patients switching to nevirapine did not have a significantly higher risk of hepatotoxicity or rash when stratified by gender and CD4 cell count, although small differences may have gone undetected because of the sample size limitation.

Publication types

  • Meta-Analysis

MeSH terms

  • Adult
  • Anti-HIV Agents / toxicity*
  • CD4 Lymphocyte Count
  • Chemical and Drug Induced Liver Injury*
  • Drug Therapy, Combination
  • Exanthema / chemically induced*
  • Exanthema / epidemiology
  • Female
  • HIV Infections / drug therapy*
  • HIV Infections / immunology*
  • HIV-1
  • Humans
  • Liver Diseases / epidemiology
  • Male
  • Middle Aged
  • Nevirapine / toxicity*
  • Randomized Controlled Trials as Topic
  • Sex Factors
  • Viral Load

Substances

  • Anti-HIV Agents
  • Nevirapine