Interleukin-13 displaying retargeted oncolytic measles virus strains have significant activity against gliomas with improved specificity

Mol Ther. 2008 Sep;16(9):1556-64. doi: 10.1038/mt.2008.152. Epub 2008 Jul 29.

Abstract

The majority of glioblastoma multiforme (GBM) tumors (80%) overexpress interleukin-13 receptor alpha2 (IL-13Ralpha2), but there is no expression of IL-13Ralpha2 in normal brain. Vaccine strains of measles virus have significant antitumor activity against gliomas. We tested the hypothesis that measles virus entry could be retargeted via the IL-13Ralpha2. MV-GFP-H(AA)-IL-13 was generated from the Edmonston-NSe vaccine strain, by displaying human IL-13 at the C-terminus of the H protein, and introducing CD46 and signaling lymphocyte activation molecule (SLAM)-ablating mutations in H. The IL-13 retargeted virus showed significant cytopathic effect (CPE) against IL-13Ralpha2 overexpressing glioma lines, and lack of CPE/viral replication in normal human astrocytes and normal human fibroblasts not expressing IL-13Ralpha2. In vivo treatment of orthotopically implanted GBM12 xenografts demonstrated significant prolongation of survival in mice treated with the retargeted strain (P < 0.0001), and comparable activity between the IL-13R retargeted strain and MV-GFP (P = 0.6377). In contrast to MV-GFP-treated mice, administration of the retargeted strain in the central nervous system of measles replication-permissive Ifnar(ko) CD46 Ge mice resulted in lack of neurotoxicity. Strains of measles virus retargeted against the glioma-specific IL-13Ralpha2 receptor have comparable therapeutic efficacy, and improved specificity as compared with the unmodified measles virus strain MV-GFP in vitro and in vivo.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Blotting, Western
  • Brain Neoplasms / genetics
  • Brain Neoplasms / immunology
  • Brain Neoplasms / therapy*
  • Central Nervous System / metabolism
  • Central Nervous System / virology
  • Chlorocebus aethiops
  • Flow Cytometry
  • Genetic Therapy*
  • Glioma / genetics
  • Glioma / immunology
  • Glioma / therapy*
  • Green Fluorescent Proteins / genetics
  • Green Fluorescent Proteins / immunology
  • Humans
  • Interleukin-13 / metabolism*
  • Interleukin-13 Receptor alpha2 Subunit / genetics
  • Interleukin-13 Receptor alpha2 Subunit / therapeutic use*
  • Measles / genetics
  • Measles / immunology
  • Measles / therapy
  • Measles virus / physiology*
  • Mice
  • Mice, Inbred BALB C
  • Mice, Nude
  • Nucleocapsid Proteins / metabolism
  • Oncolytic Virotherapy*
  • Tumor Cells, Cultured
  • Vero Cells
  • Xenograft Model Antitumor Assays

Substances

  • Interleukin-13
  • Interleukin-13 Receptor alpha2 Subunit
  • Nucleocapsid Proteins
  • Green Fluorescent Proteins