Adefovir dipivoxil is effective for the treatment of cirrhotic patients with lamivudine failure

Liver Int. 2009 Mar;29(3):420-6. doi: 10.1111/j.1478-3231.2008.01867.x. Epub 2008 Sep 15.

Abstract

Background/aims: Data on the efficacy of adefovir dipivoxil (ADV) in elderly and cirrhotic patients with lamivudine-resistant (LAM-R) chronic hepatitis B are scarce. This retrospective cohort study evaluated the safety and efficacy of ADV in this specific patient population.

Methods: Sixty-eight cirrhotic LAM-R patients, of whom 19 (27.9%) were elderly (>or=65 years of age) and nine had severe disease (two post-orthotopic liver transplantation, four pre-orthotopic liver transplantation and three decompensated), with hepatitis B virus (HBV) infection received ADV. Virological and biochemical responses to the addition of ADV were analysed.

Results: At inclusion, all patients were receiving LAM; ADV was added. 75.4% of patients received a combination of LAM and ADV throughout this study for a median treatment duration of 12.6 months; the remainder received ADV with an overlap with LAM treatment for a median duration of 7.9 months. At the end of follow-up, 41.2% of patients had undetectable HBV DNA (<or=2000 copies/ml) with a median reduction of 3.4 log(10) copies/ml. Time to reach undetectable HBV DNA was dependent on baseline alanine aminotransferase (ALT) levels and HBeAg status. Normalization of serum ALT levels was observed in 55.2% (32/58) of patients. In patients who were HBeAg positive at baseline, HBeAg loss and seroconversion occurred in 23% (9/39) and 10% (4/39) respectively. No resistance mutations and no significant side effects were observed during the study period.

Conclusion: Adefovir dipivoxil provides effective and safe treatment in cirrhotic and elderly patients who failed LAM therapy.

Publication types

  • Multicenter Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenine / analogs & derivatives*
  • Adenine / therapeutic use
  • Adult
  • Aged
  • Alanine Transaminase / metabolism
  • Cohort Studies
  • Drug Resistance / physiology
  • Female
  • Genotype
  • Hepatitis B e Antigens / metabolism
  • Hepatitis B virus / genetics
  • Hepatitis B, Chronic / complications*
  • Humans
  • Lamivudine
  • Liver Cirrhosis / drug therapy*
  • Liver Cirrhosis / etiology
  • Male
  • Middle Aged
  • Organophosphonates / therapeutic use*
  • Retrospective Studies

Substances

  • Hepatitis B e Antigens
  • Organophosphonates
  • Lamivudine
  • Alanine Transaminase
  • Adenine
  • adefovir dipivoxil