Epsilon-poly-L-lysine dispersity is controlled by a highly unusual nonribosomal peptide synthetase

Nat Chem Biol. 2008 Dec;4(12):766-72. doi: 10.1038/nchembio.125. Epub 2008 Nov 9.

Abstract

Epsilon-Poly-L-lysine (epsilon-PL) consists of 25-35 L-lysine residues in isopeptide linkages and is one of only two amino acid homopolymers known in nature. Elucidating the biosynthetic mechanism of epsilon-PL should open new avenues for creating novel classes of biopolymers. Here we report the purification of an epsilon-PL synthetase (Pls; 130 kDa) and the cloning of its gene from an epsilon-PL-producing strain of Streptomyces albulus. Pls was found to be a membrane protein with adenylation and thiolation domains characteristic of the nonribosomal peptide synthetases (NRPSs). It had no traditional condensation or thioesterase domain; instead, it had six transmembrane domains surrounding three tandem soluble domains. These tandem domains iteratively catalyzed L-lysine polymerization using free L-lysine polymer (or monomer in the initial reaction) as acceptor and Pls-bound L-lysine as donor, directly yielding chains of diverse length. Thus, Pls is a new single-module NRPS having an amino acid ligase-like catalytic activity for peptide bond formation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Bacterial Proteins
  • Catalysis
  • Cloning, Molecular
  • Membrane Proteins
  • Molecular Sequence Data
  • Peptide Biosynthesis, Nucleic Acid-Independent*
  • Peptide Synthases / metabolism*
  • Polylysine / biosynthesis*
  • Protein Conformation
  • Streptomyces / enzymology*
  • Substrate Specificity

Substances

  • Bacterial Proteins
  • Membrane Proteins
  • Polylysine
  • Peptide Synthases
  • epsilon-poly-L-lysine synthethase, Streptomyces albulus

Associated data

  • GENBANK/AB385841
  • PubChem-Substance/56260873
  • PubChem-Substance/56260874
  • PubChem-Substance/56260875
  • PubChem-Substance/56260876
  • PubChem-Substance/56260877
  • PubChem-Substance/56260878
  • PubChem-Substance/56260879
  • PubChem-Substance/56260880
  • PubChem-Substance/56260881
  • PubChem-Substance/56260882
  • PubChem-Substance/56260883
  • PubChem-Substance/56260884