The acid test: the discovery of two-pore channels (TPCs) as NAADP-gated endolysosomal Ca(2+) release channels

Pflugers Arch. 2009 Sep;458(5):869-76. doi: 10.1007/s00424-009-0682-y. Epub 2009 May 28.

Abstract

In this review, we describe the background and implications of our recent discovery that two-pore channels (TPCs) comprise a novel class of calcium release channels gated by the intracellular messenger nicotinic acid adenine dinucleotide phosphate (NAADP). Their localisation to the endolysosomal system highlights a new function for these organelles as targets for NAADP-mediated Ca(2+) mobilisation. In addition, we describe how TPCs may also trigger further Ca(2+) release by coupling to the endoplasmic reticular stores through activation of IP(3) receptors and ryanodine receptors.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Calcium Channels / physiology*
  • Calcium Signaling / physiology
  • Endosomes / physiology*
  • Humans
  • Ion Channel Gating / physiology*
  • Lysosomes / physiology*
  • Models, Molecular
  • NADP / analogs & derivatives*
  • NADP / physiology
  • Phylogeny

Substances

  • Calcium Channels
  • NADP
  • NAADP