Vaccinia virus protein F1L is a caspase-9 inhibitor

J Biol Chem. 2010 Feb 19;285(8):5569-80. doi: 10.1074/jbc.M109.078113. Epub 2009 Dec 18.

Abstract

Apoptosis plays important roles in host defense, including the elimination of virus-infected cells. The executioners of apoptosis are caspase family proteases. We report that vaccinia virus-encoded F1L protein, previously recognized as anti-apoptotic viral Bcl-2 family protein, is a caspase-9 inhibitor. F1L binds to and specifically inhibits caspase-9, the apical protease in the mitochondrial cell death pathway while failing to inhibit other caspases. In cells, F1L inhibits apoptosis and proteolytic processing of caspases induced by overexpression of caspase-9 but not caspase-8. An N-terminal region of F1L preceding the Bcl-2-like fold accounts for caspase-9 inhibition and significantly contributes to the anti-apoptotic activity of F1L. Viral F1L thus provides the first example of caspase inhibition by a Bcl-2 family member; it functions both as a suppressor of proapoptotic Bcl-2 family proteins and as an inhibitor of caspase-9, thereby neutralizing two sequential steps in the mitochondrial cell death pathway.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Apoptosis / genetics
  • Caspase 8 / chemistry
  • Caspase 8 / genetics
  • Caspase 8 / metabolism
  • Caspase 9 / chemistry
  • Caspase 9 / genetics
  • Caspase 9 / metabolism
  • Caspase Inhibitors*
  • Cattle
  • HeLa Cells
  • Humans
  • Mitochondria / chemistry
  • Mitochondria / genetics
  • Mitochondria / metabolism
  • Protein Binding / physiology
  • Protein Structure, Tertiary / genetics
  • Proto-Oncogene Proteins c-bcl-2 / chemistry
  • Proto-Oncogene Proteins c-bcl-2 / genetics
  • Proto-Oncogene Proteins c-bcl-2 / metabolism*
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / genetics
  • Recombinant Proteins / metabolism
  • Vaccinia virus / chemistry
  • Vaccinia virus / genetics
  • Vaccinia virus / metabolism*
  • Viral Proteins / chemistry
  • Viral Proteins / genetics
  • Viral Proteins / metabolism*

Substances

  • Caspase Inhibitors
  • F1L protein, vaccinia virus
  • Proto-Oncogene Proteins c-bcl-2
  • Recombinant Proteins
  • Viral Proteins
  • CASP8 protein, human
  • CASP9 protein, human
  • Caspase 8
  • Caspase 9