Etravirine limits the emergence of darunavir and other protease inhibitor resistance-associated mutations in the DUET trials

AIDS. 2010 Mar 27;24(6):921-4. doi: 10.1097/QAD.0b013e328336ac2a.

Abstract

Etravirine is a recently approved nonnucleoside reverse transcriptase inhibitor. The ability of etravirine to limit the emergence of resistance to protease inhibitors, and specifically to darunavir, was investigated in the subset of treatment-experienced patients with virologic rebound in the phase III DUET trials. Of those experiencing rebound, fewer etravirine-treated than placebo-treated patients developed mutations associated with resistance to protease inhibitors in general and to darunavir in particular, and more patients in the etravirine than the placebo-group maintained baseline darunavir susceptibility at endpoint.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antiretroviral Therapy, Highly Active
  • Drug Resistance, Multiple, Viral / drug effects*
  • Drug Resistance, Multiple, Viral / genetics
  • HIV Infections / drug therapy*
  • HIV Infections / genetics
  • HIV-1 / drug effects*
  • HIV-1 / genetics
  • Humans
  • Mutation
  • Nitriles
  • Pyridazines / pharmacology*
  • Pyrimidines
  • Reverse Transcriptase Inhibitors / pharmacology*

Substances

  • Nitriles
  • Pyridazines
  • Pyrimidines
  • Reverse Transcriptase Inhibitors
  • etravirine