Identification of a dominant negative inhibitor of human zinc finger antiviral protein reveals a functional endogenous pool and critical homotypic interactions

J Virol. 2010 May;84(9):4504-12. doi: 10.1128/JVI.02018-09. Epub 2010 Feb 24.

Abstract

The zinc finger antiviral protein (ZAP) is a host factor with potent antiviral activity when overexpressed in cells. ZAP blocks replication of the prototype alphavirus Sindbis virus (SINV) at a step at or before translation of the incoming viral genome. The mechanism of ZAP anti-SINV activity and the determinants of its antiviral function, however, have not been defined. Here, we have identified a dominant negative inhibitor of human ZAP. Rat ZAP with a cysteine-to-arginine mutation at position 88 (rZAPC88R), previously reported as a nonfunctional form of ZAP, increases SINV growth in cells. These results led us to discover a previously undetectable pool of endogenous functional ZAP within human cells. Investigation of the mechanism of dominant negative inhibition, combined with a comprehensive mutational analysis of the antiviral factor, revealed that homotypic associations are required for ZAP function in limiting SINV propagation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Substitution / genetics
  • Animals
  • Carrier Proteins / genetics*
  • Carrier Proteins / pharmacology*
  • Cell Line
  • Cells, Cultured
  • Cricetinae
  • Enzyme Inhibitors / pharmacology*
  • Humans
  • Mutant Proteins / genetics*
  • Mutant Proteins / pharmacology*
  • Mutation, Missense
  • Protein Binding
  • RNA-Binding Proteins / antagonists & inhibitors*
  • Rats
  • Sindbis Virus / growth & development*
  • Sindbis Virus / immunology
  • Viral Load

Substances

  • Carrier Proteins
  • Enzyme Inhibitors
  • Mutant Proteins
  • RNA-Binding Proteins
  • ZC3HAV1 protein, human
  • Zc3hav1 protein, rat