Abstract
TANK/I-TRAF is a TRAF-binding protein that negatively regulates NF-kappaB activation. The underlying mechanism of this activity remains unclear. Here we show that TANK directly interacts with PLK1, a conserved cell cycle-regulated kinase. PLK1 inhibits NF-kappaB transcriptional activation induced by TNF-alpha, IL-1beta, or several activators, but not by nuclear transcription factor p65. PLK1 expression reduces the DNA-binding activity of NF-kappaB induced by TNF-alpha. Moreover, endogenous activation of PLK1 reduces the TNF-induced phosphorylation of endogenous IkappaBalpha. PLK1 is bound to NEMO (IKKgamma) through TANK to form a ternary complex in vivo. We describe a new regulatory mechanism for PLK1: PLK1 negatively regulates TNF-induced IKK activation by inhibiting the ubiquitination of NEMO. These findings reveal that the scaffold protein TANK recruits PLK1 to negatively regulate NF-kappaB activation and provide direct evidence that PLK1 is required for the repression function of TANK.
Publication types
-
Research Support, Non-U.S. Gov't
MeSH terms
-
Adaptor Proteins, Signal Transducing / metabolism*
-
Cell Cycle / drug effects
-
Cell Cycle Proteins / metabolism*
-
Cell Line
-
Cytoplasm / drug effects
-
Cytoplasm / enzymology
-
Enzyme Activation / drug effects
-
Humans
-
I-kappa B Kinase / metabolism
-
I-kappa B Proteins / metabolism
-
Mutation / genetics
-
NF-KappaB Inhibitor alpha
-
NF-kappa B / genetics*
-
NF-kappa B / metabolism
-
Phosphorylation / drug effects
-
Polo-Like Kinase 1
-
Protein Binding / drug effects
-
Protein Interaction Mapping
-
Protein Processing, Post-Translational / drug effects
-
Protein Serine-Threonine Kinases / metabolism*
-
Protein Transport / drug effects
-
Proto-Oncogene Proteins / metabolism*
-
Transcriptional Activation / drug effects
-
Transcriptional Activation / genetics*
-
Tumor Necrosis Factor-alpha / pharmacology
-
Two-Hybrid System Techniques
-
Ubiquitination / drug effects
Substances
-
Adaptor Proteins, Signal Transducing
-
Cell Cycle Proteins
-
I-kappa B Proteins
-
IKBKG protein, human
-
NF-kappa B
-
NFKBIA protein, human
-
Proto-Oncogene Proteins
-
TANK protein, human
-
Tumor Necrosis Factor-alpha
-
NF-KappaB Inhibitor alpha
-
Protein Serine-Threonine Kinases
-
TBK1 protein, human
-
I-kappa B Kinase