In vitro bioaccessibility and gut biotransformation of polyphenols present in the water-insoluble cocoa fraction

Mol Nutr Food Res. 2011 May:55 Suppl 1:S44-55. doi: 10.1002/mnfr.201000360. Epub 2011 Feb 3.

Abstract

Scope: Cocoa, especially the water-insoluble cocoa fraction (WICF), is a rich source of polyphenols. In this study, sequential in vitro digestion of the WICF with gastrointestinal enzymes as well as its bacterial fermentation in a human colonic model system were carried out to investigate bioaccessibility and biotransformation of WICF polyphenols, respectively.

Methods and results: The yield of each enzymatic digestion step and the total antioxidant capacity (TAC) were measured and solubilized phenols were characterized by MS/MS. Fermentation of WICF and the effect on the gut microbiota, SCFA production and metabolism of polyphenols was analyzed. In vitro digestion solubilized 38.6% of WICF with pronase and Viscozyme L treatments releasing 51% of the total phenols from the insoluble material. This release of phenols does not determine a reduction in the total antioxidant capacity of the digestion-resistant material. In the colonic model WICF significantly increased of bifidobacteria and lactobacilli as well as butyrate production. Flavanols were converted into phenolic acids by the microbiota following a concentration gradient resulting in high concentrations of 3-hydroxyphenylpropionic acid (3-HPP) in the last gut compartment.

Conclusion: Data showed that WICF may exert antioxidant action through the gastrointestinal tract despite its polyphenols being still bound to macromolecules and having prebiotic activity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Antioxidants / analysis
  • Bacteria / drug effects
  • Bacteria / metabolism
  • Biological Availability
  • Biotransformation
  • Cacao / chemistry*
  • Digestion
  • Fermentation*
  • Flavonoids / pharmacokinetics*
  • Gastrointestinal Tract / metabolism*
  • Gastrointestinal Tract / microbiology
  • Humans
  • Hydroxybenzoates / metabolism
  • Male
  • Metagenome
  • Phenols / pharmacokinetics*
  • Polyphenols
  • Propionates / analysis

Substances

  • 3-hydroxyphenylpropionic acid
  • Antioxidants
  • Flavonoids
  • Hydroxybenzoates
  • Phenols
  • Polyphenols
  • Propionates
  • phenolic acid