ER stress inhibits mTORC2 and Akt signaling through GSK-3β-mediated phosphorylation of rictor

Sci Signal. 2011 Feb 22;4(161):ra10. doi: 10.1126/scisignal.2001731.

Abstract

In response to environmental cues, cells coordinate a balance between anabolic and catabolic pathways. In eukaryotes, growth factors promote anabolic processes and stimulate cell growth, proliferation, and survival through activation of the phosphoinositide 3-kinase (PI3K)-Akt pathway. Akt-mediated phosphorylation of glycogen synthase kinase-3β (GSK-3β) inhibits its enzymatic activity, thereby stimulating glycogen synthesis. We show that GSK-3β itself inhibits Akt by controlling the mammalian target of rapamycin complex 2 (mTORC2), a key activating kinase for Akt. We found that during cellular stress, GSK-3β phosphorylated the mTORC2 component rictor at serine-1235, a modification that interfered with the binding of Akt to mTORC2. The inhibitory effect of GSK-3β on mTORC2-Akt signaling and cell proliferation was eliminated by blocking phosphorylation of rictor at serine-1235. Thus, in response to cellular stress, GSK-3β restrains mTORC2-Akt signaling by specifically phosphorylating rictor, thereby balancing the activities of GSK-3β and Akt, two opposing players in glucose metabolism.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Carrier Proteins / chemistry
  • Carrier Proteins / metabolism*
  • Endoplasmic Reticulum / metabolism*
  • Enzyme Activation
  • Glycogen Synthase Kinase 3 / metabolism*
  • Glycogen Synthase Kinase 3 beta
  • Humans
  • Phosphorylation
  • Proto-Oncogene Proteins c-akt / metabolism*
  • Rapamycin-Insensitive Companion of mTOR Protein
  • Serine / metabolism
  • Stress, Physiological*
  • Substrate Specificity
  • Transcription Factors / metabolism*

Substances

  • CRTC2 protein, human
  • Carrier Proteins
  • RICTOR protein, human
  • Rapamycin-Insensitive Companion of mTOR Protein
  • Transcription Factors
  • Serine
  • GSK3B protein, human
  • Glycogen Synthase Kinase 3 beta
  • Proto-Oncogene Proteins c-akt
  • Glycogen Synthase Kinase 3