Anthraquinones from Morinda officinalis roots enhance adipocyte differentiation in 3T3-L1 cells

Nat Prod Res. 2012;26(18):1750-4. doi: 10.1080/14786419.2011.608676. Epub 2011 Oct 18.

Abstract

To search for anti-diabetic and insulin-sensitising natural products, the effect on adipocyte differentiation was investigated by assessing fat accumulation in 3T3-L1 preadipocytes using Oil Red O staining. Fractionation and separation of n-hexane and CHCl₃ fractions of Morinda officinalis (Rubiaceae) using several chromatographic methods led to the isolation of three anthraquinones, 1,2-dimethoxyanthraquinone (1), alizarin-2-methyl ether (2) and rubiadin-1-methyl ether (3). Among them, alizarin-2-methyl ether (2) showed the strongest enhancing activity, followed by rubiadin-1-methyl ether (3) and 1,2-dimethoxyanthraquinone (1). At a concentration of 100 µM, alizarin-2-methyl ether (2) enhanced adipocyte differentiation by up to 131% (compared to insulin-treated cells). Thus, these compounds could be beneficial in the treatment of diabetes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3T3-L1 Cells
  • Adipocytes / cytology*
  • Adipocytes / drug effects*
  • Animals
  • Anthraquinones / chemistry*
  • Anthraquinones / pharmacology*
  • Cell Differentiation / drug effects*
  • Mice
  • Morinda / chemistry*
  • Plant Roots / chemistry*

Substances

  • Anthraquinones