CCR5 blockade is well tolerated and induces changes in the tissue distribution of CCR5+ and CD25+ T cells in healthy, SIV-uninfected rhesus macaques

J Med Primatol. 2012 Feb;41(1):24-42. doi: 10.1111/j.1600-0684.2011.00521.x. Epub 2011 Nov 14.

Abstract

Background: CCR5 is a main co-receptor for HIV, but also homes lymphocytes to sites of inflammation. We hypothesized that inhibition of CCR5 signaling would reduce HIV-associated chronic immune activation.

Methods: To test this hypothesis, we administered an antagonistic anti-CCR5 monoclonal antibody (HGS101) to five uninfected rhesus macaques (RMs) and monitored lymphocyte dynamics in blood and tissue.

Results: CCR5 blockade resulted in decreased levels of CCR5+ T cells in blood and, at later timepoints, in lymph nodes. Additionally, the levels of CD25+ T cells increased in lymph nodes, but decreased in blood, bone marrow, and rectal mucosa. Finally, a profile of gene expression from HGS101-treated RMs revealed a subtle, but consistent, in vivo signature of CCR5 blockade that suggests a mild immune-modulatory effect.

Conclusions: Treatment with anti-CCR5 antibody induces changes in the tissue distribution of CCR5+ and CD25+ T cells that may impact on the overall levels of immune activation during HIV and SIV infection.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Antibodies, Monoclonal / pharmacology*
  • CCR5 Receptor Antagonists*
  • Flow Cytometry / veterinary
  • Immunophenotyping / veterinary
  • Interleukin-2 Receptor alpha Subunit / immunology*
  • Longitudinal Studies
  • Lymphoid Tissue / immunology*
  • Macaca mulatta / blood
  • Macaca mulatta / immunology*
  • Oligonucleotide Array Sequence Analysis
  • RNA / chemistry
  • RNA / genetics
  • Receptors, CCR5 / immunology
  • Reverse Transcriptase Polymerase Chain Reaction
  • Simian Acquired Immunodeficiency Syndrome / immunology
  • Simian Immunodeficiency Virus
  • T-Lymphocytes / immunology*

Substances

  • Antibodies, Monoclonal
  • CCR5 Receptor Antagonists
  • Interleukin-2 Receptor alpha Subunit
  • Receptors, CCR5
  • RNA