Stromal control of cystine metabolism promotes cancer cell survival in chronic lymphocytic leukaemia

Nat Cell Biol. 2012 Feb 19;14(3):276-86. doi: 10.1038/ncb2432.

Abstract

Tissue stromal cells interact with leukaemia cells and profoundly affect their viability and drug sensitivity. Here we show a biochemical mechanism by which bone marrow stromal cells modulate the redox status of chronic lymphocytic leukaemia (CLL) cells and promote cellular survival and drug resistance. Primary CLL cells from patients exhibit a limited ability to transport cystine for glutathione (GSH) synthesis owing to a low expression level of Xc-transporter. In contrast, bone marrow stromal cells effectively import cystine and convert it to cysteine, which is then released into the microenvironment for uptake by CLL cells to promote GSH synthesis. The elevated level of GSH enhances leukaemia cell survival and protects them from drug-induced cytotoxicity. Furthermore, disabling this protective mechanism significantly sensitizes CLL cells to drug treatment in the stromal environment. This stromal-leukaemia interaction is critical for CLL cell survival and represents a key biochemical pathway for effectively targeting leukaemia cells to overcome drug resistance in vivo.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / pharmacology
  • Blotting, Western
  • Bone Marrow Cells / cytology
  • Bone Marrow Cells / metabolism*
  • Cell Communication
  • Cell Line
  • Cell Survival / drug effects
  • Coculture Techniques
  • Culture Media, Conditioned / chemistry
  • Culture Media, Conditioned / metabolism
  • Culture Media, Conditioned / pharmacology
  • Cysteine / metabolism
  • Cystine / metabolism*
  • Drug Resistance, Neoplasm
  • Flow Cytometry
  • Glutathione / biosynthesis*
  • Humans
  • Leukemia, Lymphocytic, Chronic, B-Cell / metabolism
  • Leukemia, Lymphocytic, Chronic, B-Cell / pathology
  • Molecular Weight
  • Organoplatinum Compounds / pharmacology
  • Oxaliplatin
  • Reactive Oxygen Species / metabolism
  • Stromal Cells / cytology
  • Stromal Cells / metabolism*
  • Tumor Cells, Cultured
  • Vidarabine / analogs & derivatives
  • Vidarabine / pharmacology

Substances

  • Antineoplastic Agents
  • Culture Media, Conditioned
  • Organoplatinum Compounds
  • Reactive Oxygen Species
  • Oxaliplatin
  • Cystine
  • Vidarabine
  • Glutathione
  • Cysteine
  • fludarabine