Signal transducer and activator of transcription 3 (STAT3) protein suppresses adenoma-to-carcinoma transition in Apcmin/+ mice via regulation of Snail-1 (SNAI) protein stability

J Biol Chem. 2012 May 25;287(22):18182-9. doi: 10.1074/jbc.M111.328831. Epub 2012 Apr 10.

Abstract

STAT3 was recently reported to suppress tumor invasion in Apc(min)(/+) mice. We investigated the mechanisms by which STAT3 inhibits intestinal epithelial tumors using Apc(min)(/+)/Stat3(IEC-KO) mice (intestinal epithelial cell (IEC)-specific deletion of STAT3 in the Apc(min)(/+) background) to determine the role of STAT3 in carcinogenesis in vivo as well as colorectal cancer cell lines in vitro. To inhibit invasion of IEC tumors, STAT3 functions as a molecular adaptor rather than a transcription factor. Accordingly, the tumors in Apc(min)(/+)/Stat3(IEC-KO) mice undergo adenoma-to-carcinoma transition and acquire an invasive phenotype. Similarly, STAT3 knockdown in a colorectal cell line enhances IEC invasion. We demonstrate that STAT3 down-regulates SNAI (Snail-1) expression levels and hence suppresses epithelial-mesenchymal transition of colorectal cancer cells. Mechanistically, STAT3 facilitates glycogen synthase kinase (GSK) 3β-mediated degradation of SNAI by regulating phosphorylation of GSK3β. Our data identified a new role for STAT3 in the adenoma-to-carcinoma sequence of intestinal tumors.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenoma / pathology*
  • Animals
  • Base Sequence
  • Carcinoma / pathology*
  • Cell Proliferation
  • DNA Primers
  • Down-Regulation
  • Epithelial-Mesenchymal Transition
  • Genes, APC*
  • Intestinal Neoplasms / pathology
  • Mice
  • Mice, Knockout
  • Polymerase Chain Reaction
  • RNA, Small Interfering
  • STAT3 Transcription Factor / genetics
  • STAT3 Transcription Factor / physiology*
  • Snail Family Transcription Factors
  • Transcription Factors / genetics
  • Transcription Factors / physiology*

Substances

  • DNA Primers
  • RNA, Small Interfering
  • STAT3 Transcription Factor
  • Snai1 protein, mouse
  • Snail Family Transcription Factors
  • Stat3 protein, mouse
  • Transcription Factors