Chronic epithelial NF-κB activation accelerates APC loss and intestinal tumor initiation through iNOS up-regulation

Proc Natl Acad Sci U S A. 2012 Aug 28;109(35):14007-12. doi: 10.1073/pnas.1211509109. Epub 2012 Aug 14.

Abstract

The role of NF-κB activation in tumor initiation has not been thoroughly investigated. We generated Ikkβ(EE)(IEC) transgenic mice expressing constitutively active IκB kinase β (IKKβ) in intestinal epithelial cells (IECs). Despite absence of destructive colonic inflammation, Ikkβ(EE)(IEC) mice developed intestinal tumors after a long latency. However, when crossed to mice with IEC-specific allelic deletion of the adenomatous polyposis coli (Apc) tumor suppressor locus, Ikkβ(EE)(IEC) mice exhibited more β-catenin(+) early lesions and visible small intestinal and colonic tumors relative to Apc(+/ΔIEC) mice, and their survival was severely compromised. IEC of Ikkβ(EE)(IEC) mice expressed high amounts of inducible nitric oxide synthase (iNOS) and elevated DNA damage markers and contained more oxidative DNA lesions. Treatment of Ikkβ(EE)(IEC)/Apc(+/ΔIEC) mice with an iNOS inhibitor decreased DNA damage markers and reduced early β-catenin(+) lesions and tumor load. The results suggest that persistent NF-κB activation in IEC may accelerate loss of heterozygocity by enhancing nitrosative DNA damage.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenomatous Polyposis Coli Protein / metabolism*
  • Animals
  • Colitis / metabolism
  • Colitis / pathology
  • Colorectal Neoplasms / genetics
  • Colorectal Neoplasms / immunology
  • Colorectal Neoplasms / metabolism*
  • Colorectal Neoplasms / pathology
  • DNA Damage / physiology
  • Epithelial Cells / metabolism
  • Female
  • I-kappa B Kinase / genetics*
  • I-kappa B Kinase / metabolism*
  • Intestinal Mucosa / immunology
  • Intestinal Mucosa / metabolism
  • Intestinal Mucosa / pathology
  • Loss of Heterozygosity / physiology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Transgenic
  • NF-kappa B / metabolism*
  • Nitric Oxide Synthase Type II / metabolism*
  • Reactive Nitrogen Species / metabolism
  • Stem Cells / cytology
  • beta Catenin / metabolism

Substances

  • Adenomatous Polyposis Coli Protein
  • CTNNB1 protein, mouse
  • NF-kappa B
  • Reactive Nitrogen Species
  • beta Catenin
  • Nitric Oxide Synthase Type II
  • Nos2 protein, mouse
  • I-kappa B Kinase