Anti-amyloid-β-mediated positron emission tomography imaging in Alzheimer's disease mouse brains

PLoS One. 2012;7(12):e51958. doi: 10.1371/journal.pone.0051958. Epub 2012 Dec 21.

Abstract

Antibody-mediated imaging of amyloid β (Aβ) in Alzheimer's disease (AD) offers a promising strategy to detect and monitor specific Aβ species, such as oligomers, that have important pathological and therapeutic relevance. The major current limitation of antibodies as a diagnostic and imaging device is poor blood-brain-barrier permeability. A classical anti-Aβ antibody, 6E10, is modified with 10 kDa polyethylene glycol (PEG) and a positron emitting isotope, Copper-64 (t(½) = 12.7 h), and intravenously delivered to the TgCRND8 mouse model of Alzheimer's disease. Modification of 6E10 with PEG (6E10-PEG) increases accumulation of 6E10 in brain tissue in both TgCRND8 and wild type control animals. 6E10-PEG differentiates TgCRND8 animals from wild type controls using positron emission tomography (PET) and provides a framework for using antibodies to detect pathology using non-invasive medical imaging techniques.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alzheimer Disease / diagnosis
  • Alzheimer Disease / metabolism*
  • Amyloid beta-Peptides / immunology
  • Amyloid beta-Peptides / metabolism*
  • Animals
  • Antibodies / chemistry
  • Antibodies / immunology
  • Antibodies / pharmacology
  • Blood-Brain Barrier / pathology
  • Brain / metabolism*
  • Brain / pathology*
  • Disease Models, Animal
  • Humans
  • Immunoglobulin G / chemistry
  • Immunoglobulin G / immunology
  • Immunoglobulin G / pharmacology
  • Mice
  • Mice, Transgenic
  • Osmotic Pressure
  • Positron-Emission Tomography*
  • Protein Binding
  • Rabbits

Substances

  • Amyloid beta-Peptides
  • Antibodies
  • Immunoglobulin G