Fibroblast growth factor 2 inhibits bone morphogenetic protein 9-induced osteogenic differentiation of mesenchymal stem cells by repressing Smads signaling and subsequently reducing Smads dependent up-regulation of ALK1 and ALK2

Int J Biochem Cell Biol. 2013 Aug;45(8):1639-46. doi: 10.1016/j.biocel.2013.05.005. Epub 2013 May 13.

Abstract

Understanding the interactions between growth factors and bone morphogenic proteins (BMPs) signaling remains a crucial issue to optimize the use of mesenchymal stem cells (MSCs) and BMPs in bone tissue engineering. BMP9 is highly capable of promoting osteogenic differentiation of MSCs. Fibroblast growth factor 2 (FGF2) is abundantly secreted during the healing process of fractures or in surgery bone sites. Herein, we explore the detail effect of FGF2 on BMP9-induced osteogenic differentiation of MSCs. It was found that FGF2 inhibited BMP9-induced osteogenic differentiation by blocking BMP9-induced Smads signaling and subsequently reducing Smads dependent up-regulation of ALK1 and ALK2 in MSCs. This effect was rescued by exogenous expression of ALK1 and ALK2, which are proved to be receptors for BMP9. Our results discovered a clue to explain the mechanism involved in the inhibitory effect of FGF2 on BMP9-induced osteogenic differentiation of MSCs. This crosstalk between FGF2 and BMP9 should be emphasized in the future use of BMP9 in therapeutic purpose of fracture repair.

Keywords: Bone morphogenic proteins 9; Fibroblast growth factor 2; Mesenchymal stem cells; Osteogenic differentiation; Smads.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Activin Receptors, Type I / metabolism*
  • Activin Receptors, Type II
  • Alkaline Phosphatase / metabolism
  • Animals
  • Cell Differentiation* / drug effects
  • Cell Line
  • Cell Proliferation / drug effects
  • Core Binding Factor Alpha 1 Subunit / metabolism
  • Fibroblast Growth Factor 2 / metabolism*
  • Growth Differentiation Factor 2 / metabolism*
  • Growth Differentiation Factor 2 / pharmacology
  • Mesenchymal Stem Cells / cytology*
  • Mesenchymal Stem Cells / drug effects
  • Mesenchymal Stem Cells / enzymology
  • Mice
  • Osteogenesis* / drug effects
  • Signal Transduction / drug effects
  • Smad Proteins / metabolism*
  • Up-Regulation / drug effects

Substances

  • Core Binding Factor Alpha 1 Subunit
  • Growth Differentiation Factor 2
  • Runx2 protein, mouse
  • Smad Proteins
  • Fibroblast Growth Factor 2
  • Activin Receptors, Type I
  • Activin Receptors, Type II
  • Acvr1 protein, mouse
  • Acvrl1 protein, mouse
  • Alkaline Phosphatase