Molecular analysis of patients with polycythemia vera or essential thrombocythemia receiving pegylated interferon α-2a

Blood. 2013 Aug 8;122(6):893-901. doi: 10.1182/blood-2012-07-442012. Epub 2013 Jun 19.

Abstract

Pegylated interferon α-2a (PEG-IFN-α-2a) has previously been shown to induce hematologic and molecular responses in patients with polycythemia vera (PV) or essential thrombocythemia (ET). Here we present a follow-up of a phase 2 trial with PEG-IFN-α-2a treatment in 43 PV and 40 ET patients with detailed molecular analysis. After a median follow-up of 42 months, complete hematologic response was achieved in 76% of patients with PV and 77% of those with ET. This was accompanied by complete molecular response (CMR) (ie, undetectable JAK2V617F) in 18% and 17%, of PV and ET patients, respectively. Serial sequencing of TET2, ASXL1, EZH2, DNMT3A, and IDH1/2 revealed that patients failing to achieve CMR had a higher frequency of mutations outside the Janus kinase-signal transducer and activator of transcription pathway and were more likely to acquire new mutations during therapy. Patients with both JAK2V617F and TET2 mutations at therapy onset had a higher JAK2V617F mutant allele burden and a less significant reduction in JAK2V617F allele burden compared with JAK2 mutant/TET2 wild-type patients. These data demonstrate that PEG-IFN-α-2a induces sustained CMR in a subset of PV or ET patients, and that genotypic context may influence clinical and molecular response to PEG-IFN-α-2a.

Publication types

  • Clinical Trial, Phase II
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • DNA Mutational Analysis
  • DNA-Binding Proteins / genetics*
  • Dioxygenases
  • Epigenesis, Genetic
  • Female
  • Follow-Up Studies
  • Genotype
  • Humans
  • Interferon-alpha / therapeutic use*
  • Janus Kinase 2 / genetics*
  • Male
  • Middle Aged
  • Polycythemia Vera / genetics*
  • Polycythemia Vera / therapy
  • Polyethylene Glycols / therapeutic use*
  • Prospective Studies
  • Proto-Oncogene Proteins / genetics*
  • Recombinant Proteins / therapeutic use
  • Remission Induction
  • Thrombocythemia, Essential / genetics*
  • Thrombocythemia, Essential / therapy
  • Treatment Outcome
  • Young Adult

Substances

  • DNA-Binding Proteins
  • Interferon-alpha
  • Proto-Oncogene Proteins
  • Recombinant Proteins
  • Polyethylene Glycols
  • Dioxygenases
  • TET2 protein, human
  • JAK2 protein, human
  • Janus Kinase 2
  • peginterferon alfa-2a