Amelioration of autoimmune arthritis by naringin through modulation of T regulatory cells and Th1/Th2 cytokines

Cell Immunol. 2014 Feb;287(2):112-20. doi: 10.1016/j.cellimm.2014.01.001. Epub 2014 Jan 13.

Abstract

Naringin, a well-known flavanone glycoside found in grapefruit and other citrus fruits, was determined to be an effective anti-inflammatory compound. We investigated the effect of naringin on the key mediators of arthritic inflammation, namely T cell subsets, CD4(+)GITR(+) expressing cells, CD4(+)CD25(+)Foxp3(+) (Treg), Th1/Th2 cytokines and inflammatory mediators. We treated Balb/c mice (p.o.) with naringin (20, 40 and 80 mg/kg) for 14 days. Compared with the vehicle-treated and arthritic-control mice, the naringin treatment demonstrated a considerable decrease in the level of T cells, CD4(+)GITR(+), Th1 cytokine and inflammatory mediator expressions. In contrast, naringin treatment resulted in significantly up-regulated Treg and Th2 cytokine levels. Therefore, the naringin-induced inhibition of the T cells, various pro-inflammatory cytokines and inflammatory mediators that facilitate cellular infiltration into the joints might have contributed to its anti-arthritic activity. Our data suggest that naringin diminished the AIA in mice and it could be a potential alternative/adjunct treatment for RA.

Keywords: Adjuvant induced arthritis; Inflammatory mediators; Mouse model; Naringin; T cell subsets; Treg cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / therapeutic use*
  • Arthritis / immunology
  • Arthritis / therapy*
  • Autoimmune Diseases / immunology
  • Autoimmune Diseases / therapy*
  • CD4 Antigens / metabolism
  • Cells, Cultured
  • Citrus paradisi / chemistry*
  • Cytokines / metabolism
  • Disease Progression
  • Female
  • Flavanones / therapeutic use*
  • Forkhead Transcription Factors / metabolism
  • Glucocorticoid-Induced TNFR-Related Protein / metabolism
  • Inflammation Mediators / metabolism
  • Interleukin-2 Receptor alpha Subunit / metabolism
  • Mice
  • Mice, Inbred BALB C
  • T-Lymphocyte Subsets / drug effects*
  • T-Lymphocyte Subsets / immunology
  • T-Lymphocytes, Regulatory / drug effects*
  • T-Lymphocytes, Regulatory / immunology
  • Th1-Th2 Balance

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • CD4 Antigens
  • Cytokines
  • Flavanones
  • Forkhead Transcription Factors
  • Foxp3 protein, mouse
  • Glucocorticoid-Induced TNFR-Related Protein
  • Inflammation Mediators
  • Interleukin-2 Receptor alpha Subunit
  • Tnfrsf18 protein, mouse
  • naringin