Structural basis for Klf4 recognition of methylated DNA

Nucleic Acids Res. 2014 Apr;42(8):4859-67. doi: 10.1093/nar/gku134. Epub 2014 Feb 11.

Abstract

Transcription factor Krüppel-like factor 4 (Klf4), one of the factors directing cellular reprogramming, recognizes the CpG dinucleotide (whether methylated or unmodified) within a specific G/C-rich sequence. The binding affinity of the mouse Klf4 DNA-binding domain for methylated DNA is only slightly stronger than that for an unmodified oligonucleotide. The structure of the C-terminal three Krüppel-like zinc fingers (ZnFs) of mouse Klf4, in complex with fully methylated DNA, was determined at 1.85 Å resolution. An arginine and a glutamate interact with the methyl group. By comparison with two other recently characterized structures of ZnF protein complexes with methylated DNA, we propose a common principle of recognition of methylated CpG by C2H2 ZnF proteins, which involves a spatially conserved Arg-Glu pair.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Arginine / chemistry
  • CpG Islands
  • DNA Methylation*
  • Glutamic Acid / chemistry
  • Kruppel-Like Factor 4
  • Kruppel-Like Transcription Factors / chemistry*
  • Kruppel-Like Transcription Factors / metabolism
  • Mice
  • Molecular Sequence Data
  • Protein Binding
  • Sequence Alignment
  • Transcription Factors / chemistry

Substances

  • Klf4 protein, mouse
  • Kruppel-Like Factor 4
  • Kruppel-Like Transcription Factors
  • Transcription Factors
  • Glutamic Acid
  • Arginine

Associated data

  • PDB/4M9E