Regiospecific C-N photocyclization of 2-styrylquinolines

J Org Chem. 2014 Jun 20;79(12):5533-7. doi: 10.1021/jo500696n. Epub 2014 May 30.

Abstract

Regiospecific C-N photocyclization of 2-styrylquinolines resulting in formation of potentially biologically active quino[1,2-a]quinolizinium derivatives was investigated. The presence of strong electron-donating groups in the phenyl ring reveals to be a crucial factor managing photocyclization effectiveness. Introduction of a crown ether moiety allows changing the photoreaction parameters by means of complexation with Mg(ClO4)2.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Crown Ethers / chemistry*
  • Cyclization
  • Electrons
  • Magnesium Compounds / chemistry*
  • Perchlorates / chemistry*
  • Photochemical Processes
  • Quinazolines / chemical synthesis*
  • Quinazolines / chemistry*
  • Quinolines / chemistry*

Substances

  • Crown Ethers
  • Magnesium Compounds
  • Perchlorates
  • Quinazolines
  • Quinolines
  • styrylquinoline
  • magnesium perchlorate