Skp2-macroH2A1-CDK8 axis orchestrates G2/M transition and tumorigenesis

Nat Commun. 2015 Mar 30:6:6641. doi: 10.1038/ncomms7641.

Abstract

Understanding the mechanism by which cell growth, migration, polyploidy, and tumorigenesis are regulated may provide important therapeutic strategies for cancer therapy. Here we identify the Skp2-macroH2A1 (mH2A1)-cyclin-dependent kinase 8 (CDK8) axis as a critical pathway for these processes, and deregulation of this pathway is associated with human breast cancer progression and patient survival outcome. We showed that mH2A1 is a new substrate of Skp2 SCF complex whose degradation by Skp2 promotes CDK8 gene and protein expression. Strikingly, breast tumour suppression on Skp2 deficiency can be rescued by mH2A1 knockdown or CDK8 restoration using mouse tumour models. We further show that CDK8 regulates p27 protein expression by facilitating Skp2-mediated p27 ubiquitination and degradation. Our study establishes a critical role of Skp2-mH2A1-CDK8 axis in breast cancer development and targeting this pathway offers a promising strategy for breast cancer therapy.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Breast Neoplasms / metabolism*
  • Carcinogenesis / genetics*
  • Carcinoma / metabolism*
  • Cell Line, Tumor
  • Cyclin-Dependent Kinase 8 / metabolism*
  • Cyclin-Dependent Kinase Inhibitor p27 / metabolism
  • Fibroblasts
  • G2 Phase Cell Cycle Checkpoints / genetics*
  • Histones / metabolism*
  • Humans
  • Mice
  • Mice, Knockout
  • S-Phase Kinase-Associated Proteins / genetics*
  • S-Phase Kinase-Associated Proteins / metabolism
  • SKP Cullin F-Box Protein Ligases / metabolism
  • Ubiquitination

Substances

  • Histones
  • S-Phase Kinase-Associated Proteins
  • macroH2A histone
  • Cyclin-Dependent Kinase Inhibitor p27
  • SKP Cullin F-Box Protein Ligases
  • CDK8 protein, human
  • Cdk8 protein, mouse
  • Cyclin-Dependent Kinase 8

Associated data

  • GEO/GSE23064