Lopinavir and atazanavir in pregnancy: comparable infant outcomes, virological efficacies and preterm delivery rates

HIV Med. 2016 Jan;17(1):28-35. doi: 10.1111/hiv.12277. Epub 2015 Jul 22.

Abstract

Objectives: The aim of the study was to identify differences in infant outcomes, virological efficacy, and preterm delivery (PTD) outcome between women exposed to lopinavir/ritonavir (LPV/r) and those exposed to atazanavir/ritonavir (ATV/r).

Methods: A retrospective case note review was carried out. The case notes of 493 women who conceived while on LPV/r or ATV/r or initiated LPV/r or ATV/r during pregnancy and who delivered between 1 September 2007 and 30 August 2012 were reviewed. Data collected included demographics, antiretroviral use, HIV markers, and pregnancy and infant outcomes. Infant outcomes, virological efficacies and PTD rates for LPV/r and ATV/r were compared.

Results: A total of 306 women received LPV/r (82 conceiving while on the drug and 224 commencing it post-conception) and 187 received ATV/r (96 conceiving while on the drug and 91 commencing it post-conception). Comparing the two protease inhibitors (PIs), viral suppression rates were similar and, in women starting antiretroviral therapy (ART) post-conception, the median times to first undetectable HIV viral load were not significantly different (P = 0.64). PTD rates did not differ by therapy overall (ATV/r, 13%; LPV/r, 14%) or when considering the timing of first exposure (conceiving on ART, P = 0.81; commencing ART in pregnancy, P = 0.08). Poor fetal outcomes were very uncommon. There were two transmissions, giving a mother-to-child transmission (MTCT) rate of 0.4% (95% confidence interval 0.05-1.5%).

Conclusions: Both ART regimens were well tolerated and successful in preventing MTCT. No significant differences in tolerability or in pregnancy or infant outcomes were observed, which supports the provision of a choice of PI in pregnancy.

Keywords: HIV; antiretroviral therapy; atazanavir; lopinavir; pregnancy; preterm delivery; protease inhibitor.

Publication types

  • Comparative Study

MeSH terms

  • Adolescent
  • Adult
  • Atazanavir Sulfate / administration & dosage*
  • Atazanavir Sulfate / pharmacology
  • Drug Combinations
  • Drug Therapy, Combination
  • Female
  • HIV Infections / drug therapy*
  • HIV Protease Inhibitors / administration & dosage*
  • HIV Protease Inhibitors / pharmacology
  • Humans
  • Infant
  • Infant, Newborn
  • Lopinavir / administration & dosage*
  • Lopinavir / pharmacology
  • Middle Aged
  • Pregnancy
  • Pregnancy Outcome / epidemiology
  • Premature Birth / epidemiology*
  • Premature Birth / etiology
  • Retrospective Studies
  • Ritonavir / administration & dosage*
  • Ritonavir / pharmacology
  • Treatment Outcome
  • Viral Load / drug effects*
  • Young Adult

Substances

  • Drug Combinations
  • HIV Protease Inhibitors
  • lopinavir-ritonavir drug combination
  • Lopinavir
  • Atazanavir Sulfate
  • Ritonavir