Tauroursodeoxycholate improves 2,4,6-trinitrobenzenesulfonic acid-induced experimental acute ulcerative colitis in mice

Int Immunopharmacol. 2016 Jul:36:271-276. doi: 10.1016/j.intimp.2016.04.037. Epub 2016 May 12.

Abstract

Ulcerative colitis is a chronic nonspecific inflammatory disease of unknown cause. The aim of this study was to evaluate the anti-inflammatory effect of tauroursodeoxycholate in 2, 4, 6-trinitrobenzenesulfonic acid-induced experimental colitis in mice. After the induction of colitis for 24h, the mice were administrated orally with tauroursodeoxycholate (20, 40 and 60mg/kg) and sulfasalazine (500mg/kg) by gavage for 7 consecutive days. The inhibition effects were evaluated by the body of weight change, survival rate, macroscopical and histological evaluations. Besides, myeloperoxidase (MPO) activity, interleukin (IL)-1β, interferon (IFN)-γ and tumour necrosis factor-α (TNF-α) in colon tissue were also determined by enzyme-linked immunosorbent assay. Treatment with different doses of tauroursodeoxycholate (20, 40 and 60mg/kg) significantly improved the body weight change, decreased the macroscopic and histopathological scores. Compared with the model group, the accumulation of MPO activity, the colonic tissue levels of IL-1β, IFN-γ and TNF-α were significantly reduced in the tauroursodeoxycholate treated groups. Moreover, tauroursodeoxycholate assuaged the symptoms of colitis. These results suggested that tauroursodeoxycholate has an anti-inflammatory effect in TNBS-induced ulcerative colitis in mice.

Keywords: Cytokines; Tauroursodeoxycholate; Trinitrobenzenesulfonic acid; Ulcerative colitis.

MeSH terms

  • Acute Disease
  • Administration, Oral
  • Animals
  • Anti-Inflammatory Agents / therapeutic use*
  • Body Weight / drug effects
  • Colitis, Ulcerative / chemically induced
  • Colitis, Ulcerative / drug therapy*
  • Colon / drug effects*
  • Colon / metabolism
  • Colon / pathology
  • Disease Models, Animal
  • Humans
  • Interferon-gamma / metabolism
  • Interleukin-1beta / metabolism
  • Male
  • Mice
  • Mice, Inbred BALB C
  • Peroxidase / metabolism
  • Taurochenodeoxycholic Acid / therapeutic use*
  • Trinitrobenzenesulfonic Acid
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Anti-Inflammatory Agents
  • Interleukin-1beta
  • Tumor Necrosis Factor-alpha
  • Taurochenodeoxycholic Acid
  • ursodoxicoltaurine
  • Interferon-gamma
  • Trinitrobenzenesulfonic Acid
  • Peroxidase