Effect of Iron Chelation Therapy on Glucose Metabolism in Non-Transfusion-Dependent Thalassaemia

Acta Haematol. 2017;137(1):20-26. doi: 10.1159/000450673. Epub 2016 Nov 12.

Abstract

Aims: To compare insulin sensitivity, β-cell function and iron status biomarkers in non-transfusion-dependent thalassaemia (NTDT) with iron excess during pre- and post-iron chelation.

Methods: Subjects with NTDT, aged older than 10 years, with serum ferritin >300 ng/ml, were included. Iron chelation with deferasirox (10 mg/kg/day) was prescribed daily for 6 months.

Results: Ten patients with a median age of 17.4 years were enrolled. The comparison between pre- and post-chelation demonstrated significantly lower iron load: median serum ferritin (551.4 vs. 486.2 ng/ml, p = 0.047), median TIBC (211.5 vs. 233.5 µg/dl, p = 0.009) and median non-transferrin binding iron (5.5 vs. 1.4 µM, p = 0.005). All patients had a normal oral glucose tolerance test (OGTT) both pre- and post-chelation. However, fasting plasma glucose was significantly reduced after iron chelation (85.0 vs.79.5 mg/dl, p = 0.047). MRI revealed no significant changes of iron accumulation in the heart and liver after chelation, but there was a significantly lower iron load in the pancreas, assessed by higher T2* at post-chelation compared with pre-chelation (41.9 vs. 36.7 ms, p = 0.047). No adverse events were detected.

Conclusions: A trend towards improving insulin sensitivity and β-cell function as well as a reduced pancreatic iron load was observed following 6 months of iron chelation (TCTR20160523003).

Publication types

  • Clinical Trial

MeSH terms

  • Adolescent
  • Benzoates / therapeutic use*
  • Blood Glucose / metabolism
  • Blood Transfusion
  • Chelation Therapy / methods*
  • Deferasirox
  • Drug Administration Schedule
  • Fasting
  • Female
  • Ferritins / blood
  • Glucose Tolerance Test
  • Humans
  • Insulin Resistance
  • Insulin-Secreting Cells / drug effects
  • Insulin-Secreting Cells / metabolism
  • Insulin-Secreting Cells / pathology
  • Iron / metabolism*
  • Iron Chelating Agents / therapeutic use*
  • Iron Overload / diagnostic imaging
  • Iron Overload / drug therapy*
  • Iron Overload / metabolism
  • Iron Overload / pathology
  • Liver / drug effects
  • Liver / metabolism
  • Liver / pathology
  • Magnetic Resonance Imaging
  • Male
  • Myocardium / metabolism
  • Myocardium / pathology
  • Prospective Studies
  • Thalassemia / diagnostic imaging
  • Thalassemia / drug therapy*
  • Thalassemia / metabolism
  • Thalassemia / pathology
  • Treatment Outcome
  • Triazoles / therapeutic use*
  • Young Adult

Substances

  • Benzoates
  • Blood Glucose
  • Iron Chelating Agents
  • Triazoles
  • Ferritins
  • Iron
  • Deferasirox