Biocompatible Polymeric Analogues of DMSO Prepared by Atom Transfer Radical Polymerization

Biomacromolecules. 2017 Feb 13;18(2):475-482. doi: 10.1021/acs.biomac.6b01553. Epub 2017 Jan 5.

Abstract

The synthesis of a sulfoxide-based water-soluble polymer, poly(2-(methylsulfinyl)ethyl acrylate) (polyMSEA), a polymeric analogue of DMSO, by atom transfer radical polymerization (ATRP) is reported. Well-defined linear polymers were synthesized using relatively low amounts of copper catalyst (1000 or 100 ppm). Two types of star polymers were synthesized by either an "arm-first" approach or a "core-first" approach using a biodegradable β-cyclodextrin core. The glass transition temperatures of both the linear polymer (16 °C) and star polymer (32 °C) were determined by differential scanning calorimetry (DSC). The lower critical solution temperature (LCST) of poly(MSEA) was estimated to be ca. 140 °C by extrapolating the LCST of a series of copolymers with NIPAM. Cytotoxicity tests revealed that both the linear and star polymers have low toxicity, even at concentrations up to 3 mg/mL.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, N.I.H., Extramural

MeSH terms

  • Biocompatible Materials / administration & dosage*
  • Biocompatible Materials / chemistry
  • Calorimetry, Differential Scanning
  • Catalysis
  • Cell Survival / drug effects
  • Dimethyl Sulfoxide / chemistry*
  • HEK293 Cells
  • Humans
  • Polymerization
  • Polymers / administration & dosage*
  • Polymers / chemistry
  • Transition Temperature
  • Water / chemistry

Substances

  • Biocompatible Materials
  • Polymers
  • Water
  • Dimethyl Sulfoxide