Mechanistic and therapeutic perspectives for cardiac arrhythmias: beyond ion channels

Sci China Life Sci. 2017 Apr;60(4):348-355. doi: 10.1007/s11427-016-9005-6. Epub 2017 Mar 24.

Abstract

Cardiac arrhythmias are among the most common causes of death in the world. Foundational studies established the critical role of ion channel disorders in arrhythmias, yet defects in ion channels themselves, such as mutations, may not account for all arrhythmias. Despite the progress made in recent decades, the antiarrhythmic drugs currently available have limited effectiveness, and the majority of these drugs can have proarrhythmic effects. This review describes novel knowledge on cellular mechanisms that cause cardiac arrhythmias, focuses on the dysfunction of subcellular organelles and intracellular logistics, and discusses potential strategies and challenges for developing novel, safe and effective treatments for arrhythmias.

Keywords: arrhythmia; ion channel; organelle; therapy; trafficking.

Publication types

  • Review

MeSH terms

  • Anti-Arrhythmia Agents / therapeutic use*
  • Arrhythmias, Cardiac / physiopathology*
  • Arrhythmias, Cardiac / therapy*
  • Humans
  • Ion Channels / drug effects*

Substances

  • Anti-Arrhythmia Agents
  • Ion Channels