Topical application of ointment containing 0.5% green tea catechins suppresses tongue oxidative stress in 5-fluorouracil administered rats

Arch Oral Biol. 2017 Oct:82:247-255. doi: 10.1016/j.archoralbio.2017.06.025. Epub 2017 Jun 19.

Abstract

Objective: The purpose of this study was to investigate the preventive effects of topical application of green tea catechins on tongue oxidative stress induced by 5-fluorouracil (5-FU) administration in rats.

Design: Male Wistar rats (n=28, 8 weeks old) were divided into four groups of seven rats each: a negative control group (saline administration and application of ointment without green tea catechins), a positive control group (5-FU administration and application of ointment without green tea catechins), and two experimental groups (5-FU administration and application of ointment containing 0.1% or 0.5% green tea catechins). Topical application of each ointment to the ventral surface of the tongue was performed once a day for 5days. The level of 8-hydroxydeoxyguanosine (8-OHdG) was determined to evaluate oxidative stress. Fluorescence staining was also performed to confirm nuclear factor erythroid 2-related factor 2 (Nrf2) translocation to the nucleus.

Results: After the experimental period, the ratios of 8-OHdG-positive cells in the ventral tongue tissue were higher in the positive control group than in the negative control group (P<0.05). On the other hand, those in the 0.5% green tea catechin group, but not in the 0.1% green tea catechin group, were lower than the positive control group (P<0.05). In addition, Nrf2 translocation to the nucleus was greater in the 0.5% green tea catechin group than in the positive control group (P<0.05).

Conclusions: Topical application of ointment containing 0.5% green tea catechins could prevent tongue oxidative stress in 5-FU administered rats, via up-regulation of the Nrf2 signaling pathway.

Keywords: Antioxidant capacity; Chemotherapy; Green tea catechin; Oxidative stress; Tongue.

MeSH terms

  • 8-Hydroxy-2'-Deoxyguanosine
  • Administration, Topical
  • Animals
  • Antioxidants / metabolism
  • Catechin / administration & dosage
  • Catechin / pharmacology*
  • Deoxyguanosine / analogs & derivatives
  • Deoxyguanosine / metabolism
  • Fluorouracil / toxicity*
  • Male
  • NF-E2-Related Factor 2 / metabolism
  • Ointments / administration & dosage
  • Ointments / pharmacology*
  • Oxidative Stress / drug effects*
  • Rats
  • Rats, Wistar
  • Tea*
  • Tongue / drug effects*

Substances

  • Antioxidants
  • NF-E2-Related Factor 2
  • Nfe2l2 protein, mouse
  • Ointments
  • Tea
  • 8-Hydroxy-2'-Deoxyguanosine
  • Catechin
  • Deoxyguanosine
  • Fluorouracil