The Red Algae Compound 3-Bromo-4,5-dihydroxybenzaldehyde Protects Human Keratinocytes on Oxidative Stress-Related Molecules and Pathways Activated by UVB Irradiation

Mar Drugs. 2017 Aug 25;15(9):268. doi: 10.3390/md15090268.

Abstract

Skin exposure to ultraviolet B (UVB) irradiation leads to the generation of reactive oxygen species (ROS). Excessive ROS cause aging of the skin via basement membrane/extracellular matrix degradation by matrix metalloproteinases (MMPs). We recently demonstrated that 3-bromo-4,5-dihydroxybenzaldehyde (BDB), a natural compound of red algae, had a photo-protective effect against UVB-induced oxidative stress in human keratinocytes. The present study focused on the effect of BDB on UVB-irradiated photo-aging in HaCaT keratinocytes and the underlying mechanism. BDB significantly impeded MMP-1 activation and expression, and abrogated the activation of mitogen-activated protein kinases and intracellular Ca2+ level in UVB-irradiated HaCaT cells. Moreover, BDB decreased the expression levels of c-Fos and phospho-c-Jun and the binding of activator protein-1 to the MMP-1 promoter induced by UVB irradiation. These results offer evidence that BDB is potentially useful for the prevention of UVB-irradiated skin damage.

Keywords: 3-bromo-4,5-dihydroxybenzaldehyde; activator protein-1; matrix metalloproteinase-1; mitogen-activated protein kinases; ultraviolet B.

MeSH terms

  • Benzaldehydes / chemistry
  • Benzaldehydes / isolation & purification
  • Benzaldehydes / pharmacology*
  • Humans
  • JNK Mitogen-Activated Protein Kinases / drug effects
  • Keratinocytes / drug effects*
  • Matrix Metalloproteinase 1 / metabolism
  • Oxidative Stress / drug effects*
  • Proto-Oncogene Proteins c-fos / drug effects
  • Rhodophyta / chemistry*
  • Ultraviolet Rays / adverse effects*

Substances

  • 3-bromo-4,5-dihydroxybenzaldehyde
  • Benzaldehydes
  • Proto-Oncogene Proteins c-fos
  • JNK Mitogen-Activated Protein Kinases
  • MMP1 protein, human
  • Matrix Metalloproteinase 1