The receptor protein tyrosine phosphatase PTPRB negatively regulates FGF2-dependent branching morphogenesis

Development. 2017 Oct 15;144(20):3777-3788. doi: 10.1242/dev.149120. Epub 2017 Sep 4.

Abstract

PTPRB is a transmembrane protein tyrosine phosphatase known to regulate blood vessel remodelling and angiogenesis. Here, we demonstrate that PTPRB negatively regulates branching morphogenesis in the mouse mammary epithelium. We show that Ptprb is highly expressed in adult mammary stem cells and also, although at lower levels, in oestrogen receptor-positive luminal cells. During mammary development, Ptprb expression is downregulated during puberty, a period of extensive ductal outgrowth and branching. In vivo shRNA knockdown of Ptprb in the cleared mammary fat pad transplant assay resulted in smaller epithelial outgrowths with an increased branching density and also increased branching in an in vitro organoid assay. Organoid branching was dependent on stimulation by FGF2, and Ptprb knockdown in mammary epithelial cells resulted in a higher level of fibroblast growth factor receptor (FGFR) activation and ERK1/2 phosphorylation, both at baseline and following FGF2 stimulation. Therefore, PTPRB regulates branching morphogenesis in the mammary epithelium by modulating the response of the FGFR signalling pathway to FGF stimulation. Considering the importance of branching morphogenesis in multiple taxa, our findings have general importance outside mammary developmental biology.

Keywords: Branching morphogenesis; FGFR2; Mammary stem cells; Mouse; PTPRB; Terminal end bud gene expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Body Patterning
  • Epithelial Cells / cytology
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • Female
  • Fibroblast Growth Factor 2 / pharmacology*
  • Gene Expression Profiling
  • Gene Expression Regulation, Developmental
  • Green Fluorescent Proteins / metabolism
  • Mammary Glands, Animal / growth & development*
  • Mice
  • Morphogenesis*
  • Neovascularization, Physiologic
  • Oligonucleotide Array Sequence Analysis
  • Organoids / growth & development
  • Phosphorylation
  • RNA, Small Interfering / metabolism
  • Receptor-Like Protein Tyrosine Phosphatases, Class 3 / genetics
  • Receptor-Like Protein Tyrosine Phosphatases, Class 3 / metabolism*
  • Receptors, Estrogen / metabolism
  • Receptors, Fibroblast Growth Factor / metabolism
  • Signal Transduction
  • Stem Cells / cytology
  • Transgenes

Substances

  • RNA, Small Interfering
  • Receptors, Estrogen
  • Receptors, Fibroblast Growth Factor
  • Fibroblast Growth Factor 2
  • Green Fluorescent Proteins
  • Extracellular Signal-Regulated MAP Kinases
  • Ptprb protein, mouse
  • Receptor-Like Protein Tyrosine Phosphatases, Class 3