Kaempferol modulates Angiopoietin-like protein 2 expression to lessen the mastitis in mice

Pharmacol Rep. 2018 Jun;70(3):439-445. doi: 10.1016/j.pharep.2017.11.006. Epub 2017 Nov 22.

Abstract

Background: Mastitis is inflammation of a breast (or udder). Angiopoietin-like protein 2 (ANGPTL2) has been found as a key inflammatory mediator in mastitis. Purpose of this research was to investigate the mechanisms about repressing effect of kaempferol on mastitis.

Methods: Forty mice were randomly divided into 4 groups (n=10): C57BL/6J control mice, untreated murine mastitis, 10mg/kg kaempferol treated murine mastitis (ip), and 30mg/kg kaempferol treated murine mastitis (ip). Primary cultured mouse mammary epithelial cells (MMEC) were indiscriminately divided into seven groups including control group, 10mmol/L vehicle of kaempferol group, 10μmol/L kaempferol treated group, 20μg/mL LPS treated group, 1μmol/L kaempferol plus LPS treated group, 3μmol/L kaempferol plus LPS treated group, and 10μmol/L kaempferol plus LPS treated group.

Results: In murine mastitis, kaempferol (10 or 30mg/kg) treatment prevented mastitis development, decreased myeloperoxidase (MPO) production, interleukin (IL)-6 level, tumour necrosis factor-α (TNF-α) concentration, and ANGPTL2 expression. In MMEC, kaempferol (1, 3 or 10μM) reduced MPO production, TNF-α concentration, IL-6 level, and ANGPTL2 expression.

Conclusions: The results in present study show that kaempferol modulates the expression of ANGPTL2 to lessen the mastitis in mice.

Keywords: Angiopoietin-like protein 2; Kaempferol; Murine mastitis.

MeSH terms

  • Angiopoietin-Like Protein 2
  • Angiopoietin-like Proteins / metabolism*
  • Animals
  • Epithelial Cells / drug effects
  • Epithelial Cells / metabolism
  • Female
  • Inflammation / drug therapy
  • Inflammation / metabolism
  • Interleukin-6 / metabolism
  • Kaempferols / pharmacology*
  • Mastitis / drug therapy*
  • Mastitis / metabolism*
  • Mice
  • Mice, Inbred C57BL
  • Peroxidase / metabolism
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Angiopoietin-Like Protein 2
  • Angiopoietin-like Proteins
  • Angptl2 protein, mouse
  • Interleukin-6
  • Kaempferols
  • Tumor Necrosis Factor-alpha
  • kaempferol
  • Peroxidase