Acetylation blocks DNA damage-induced chromatin ADP-ribosylation

Nat Chem Biol. 2018 Sep;14(9):837-840. doi: 10.1038/s41589-018-0097-1. Epub 2018 Jul 16.

Abstract

Recent studies report serine ADP-ribosylation on nucleosomes during the DNA damage response. We unveil histone H3 serine 10 as the primary acceptor residue for chromatin ADP-ribosylation and find that specific histone acetylation marks block this activity. Our results provide a molecular explanation for the well-documented phenomenon of rapid deacetylation at DNA damage sites and support the combinatorial application of PARP and HDAC inhibitors for the treatment of PARP-dependent cancers.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • ADP-Ribosylation*
  • Acetylation
  • Chromatin / metabolism*
  • Cloning, Molecular
  • DNA / genetics
  • DNA / metabolism
  • DNA Damage*
  • Histones / genetics
  • Histones / metabolism*
  • Humans
  • Tumor Cells, Cultured

Substances

  • Chromatin
  • Histones
  • DNA